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3-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(morpholin-4-yl)benzamide
2-[(4aR,7aS)-6,6-dioxo-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
1-{2-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}piperidin-2-one
2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[1-(3-methylphenyl)piperidin-4-yl]acetamide
3-propyl-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1H-pyrazole-5-carboxamide
(2S,4R)-4-amino-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-indazol-3-yl)acetamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-cyclopropyl-N-[2-(2,4-dimethoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(2-oxopiperidin-1-yl)acetamide
(furan-3-ylmethyl)(methyl){[(2R,5S)-5-(pyridin-4-ylmethyl)oxolan-2-yl]methyl}amine
[7-chloro-5-(2-methyl-1H-imidazol-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-(1,4-dioxan-2-ylmethyl)-2-ethoxypyridine-3-carboxamide
4-{[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}morpholine
2-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
2-benzyl-8-(ethanesulfonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5-methylpiperidin-2-one
2-{1-[(2-methylphenyl)methyl]-5-[2-(pyrazin-2-yl)ethyl]-1H-1,2,4-triazol-3-yl}acetamide
1-{9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
4-(1-benzothiophene-2-carbonyl)-N-cyclohexyl-N-methylmorpholine-2-carboxamide
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[5-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
2-(3,3,4,4-tetrafluorobutyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
4-[1-butyl-5-(2-methylpyrimidin-5-yl)-1H-1,2,4-triazol-3-yl]benzamide
N-{2-methoxy-5-[3-(1H-pyrazol-4-yl)propanamido]phenyl}pentanamide
4-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1λ6-thiane-1,1-dione
4-{5-[3-(2-phenylethyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
6-[2-chloro-3-(pyrrolidin-1-ylmethyl)phenoxy]pyrazine-2-carboxamide
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(4-fluorophenyl)sulfanyl]piperidine
2-{1-methyl-4-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]piperazin-2-yl}ethan-1-ol
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-(pyridin-3-ylmethyl)pyridin-2-amine
N-{3-hydroxy-1-[4-(propan-2-yl)phenyl]propyl}-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
2-methoxy-N-(1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
1-(3-chlorophenyl)-3-methyl-5-[2-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
3-(benzyloxy)-N-(5-propyl-4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-1-(thiomorpholin-4-yl)ethan-1-one
2-(4-chlorophenyl)-4-[(3,4-dimethoxypyridin-2-yl)methyl]morpholine
2-(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-3-(pyridin-3-yl)propan-1-one
(3R,4S)-4-{4-[(1-methyl-1H-indol-2-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
4-chloro-2-methoxy-N-propyl-N-(pyridin-3-ylmethyl)benzamide
1-[4-(2-methylpropoxy)phenyl]-3-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}urea
methyl 9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-oxo-3-[2-(thiophen-2-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl (1R,3S,3aR,6aS)-1-ethyl-5-methyl-4,6-dioxo-3-(2,4,5-trimethylphenyl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-(4-butyl-2,3-dioxopiperazin-1-yl)-N-cyclopentyl-2-phenylacetamide
3-(3-chlorophenyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-phenylpropanamide
2,5-dimethyl-3-{3-[1-(2-propoxyethyl)-1H-pyrazol-3-yl]phenyl}pyrazine
2-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one