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4-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-1,3-dimethylpiperazin-2-one
2-[(3-chlorophenyl)methyl]-N-(1-methylpiperidin-4-yl)-1,3-benzoxazole-6-carboxamide
N-cyclopropyl-2-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carboxamide
2-[4-(2-methanesulfonylethyl)piperazin-1-yl]-4-(pyridin-2-yl)pyrimidine
3-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-pyrazol-5-amine
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-4-(pyridin-3-yl)pyrimidin-2-amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]propan-1-one
1-[2-(dimethylamino)ethyl]-4-{4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}pyrrolidin-2-one
methyl 3-{[4-ethyl-5-oxo-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}benzoate
N-[(1R)-2,3-dihydro-1H-inden-1-yl]imidazo[1,2-a]pyrimidine-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylpiperidine-4-carboxamide
N-cyclobutyl-2-[(3E)-pent-3-enoyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-(4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-N-methyl-2-oxo-N-phenylacetamide
2-cyclopropyl-9-(2-hydroxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-amino-6-{4-[(2-cyclohexylpyrimidin-5-yl)methyl]piperazin-1-yl}pyrimidin-4-ol
2-(4,4-dimethyl-2-oxopyrrolidin-1-yl)-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)phenyl]methyl}-3-fluoro-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-[(3-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-1-benzofuran-3-carboxamide
2-methoxy-1-[1'-(oxane-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
1-(2-methoxyethyl)-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-benzyl-N-ethyl-3-[2-(pyridin-2-yl)pyrrolidin-1-yl]propanamide
2-butyl-1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-2,5-dihydro-1H-pyrrole
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(2E)-4-methylpent-2-en-1-yl]piperidine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
1-[(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
5-(2-oxo-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(4-chlorobenzoyl)-1-[(3-methoxyphenyl)methyl]piperidine
N,3,4,7-tetramethyl-N-(quinoxalin-6-ylmethyl)-1H-indole-2-carboxamide
1-{3-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N,N-dimethyl-6-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidin-4-amine
2-acetyl-8-[(3,5-dimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(4-{4-[(4-fluorophenyl)sulfanyl]piperidine-1-carbonyl}piperidin-1-yl)-4-methylquinazoline
3-(2-oxo-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethyl)-2,3-dihydro-1H-isoindol-1-one
1-(azocan-1-yl)-3-[2-methoxy-5-({[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-phenyl-5-{1-[1-(1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}-1,2-oxazole
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxybenzoyl)piperazine
2-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-3,5-dimethyl-1H-indole
1-(3-chlorophenyl)-4-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)piperazine
4-methyl-6-[2-(trifluoromethyl)phenyl]pyrimidin-2-amine
(3S,4R)-N,N-dimethyl-1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-4-(propan-2-yl)pyrrolidin-3-amine
1-{3-[3-(2-chlorophenoxy)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
5-[4-(4-fluorophenyl)piperazin-1-yl]-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
(1-{1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-4-yl}ethyl)dimethylamine
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-5-phenylpentan-1-one
2-[2-(dimethylamino)ethyl]-9-(pyrazin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-hydroxypiperidin-1-yl)-2-[4-(4-{[(5-phenyl-1H-pyrazol-3-yl)methyl]amino}piperidin-1-yl)phenyl]ethan-1-one
2-(diethylamino)-1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}ethan-1-one
1-[(2-chloro-6-fluorophenyl)methyl]-5-({[2-(pyrrolidin-1-yl)ethyl]sulfanyl}methyl)-1H-1,2,4-triazole
N-[3-(2-ethoxyphenyl)propyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide