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N-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-methylthieno[3,2-d]pyrimidin-4-amine
4-(4-acetamidophenyl)-6-methyl-2-oxo-N-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-4-phenylbutane-1,4-dione
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-6-(propan-2-yl)pyrimidin-2-amine
2,2-difluoro-N-({1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)acetamide
N-[(3R,4S)-1-acetyl-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]pyrrolidine-1-sulfonamide
[2-(4,6-dimethylpyrimidin-2-yl)ethyl]({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-(2,6-dimethylphenyl)-9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
2-(2-fluorophenoxymethyl)-N-[(6-methylpyridin-2-yl)methyl]-1,3-oxazole-4-carboxamide
[(3S,7S)-5-(2,5-dimethylfuran-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
2,2-dimethyl-1-(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propan-1-one
2-(adamantan-1-yl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]acetamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amine
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-[2-(phenylsulfanyl)ethyl]propanamide
2-[(3-chlorophenyl)methyl]-6-(3-methoxypiperidine-1-carbonyl)-1,3-benzoxazole
5-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-chloro-4-hydroxy-N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
2-(dimethylamino)-N-methyl-N-(1-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}-2-phenylethyl)acetamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
1-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-4-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazole
2-cyclopentanecarbonyl-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decane
4-{4-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
[(3R,4S)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(4-ethoxyphenyl)methyl]pyrrolidin-3-yl]methanol
3-{1-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
2-(3-methoxyphenoxymethyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
(1S,5R)-N-(2-chlorophenyl)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
4-methoxy-2-(4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)pyrimidine
4-({[4-methyl-5-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}methyl)pyridine
N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-propyl-1,3-thiazole-4-carboxamide
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-[2-(3-methoxyphenoxy)ethyl]piperazine
5-cyclohexaneamido-1-(2-methoxyethyl)-N-[2-(4-methoxyphenyl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
{4-[2-chloro-5-(trifluoromethyl)benzoyl]-1,4-oxazepan-6-yl}methanol
5-(3-fluorophenoxymethyl)-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
4-(5-ethylthiophene-3-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
3-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1-phenylurea
N-(1,2-oxazol-3-ylmethyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-ethyl-4-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-cyclopropyl-N-[2-(3-methylthiophen-2-yl)ethyl]-1H-pyrazole-5-carboxamide
3-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridin-2-ol
2-[(2-{1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
1-(oxan-4-yl)-3-[3-(trifluoromethyl)benzoyl]piperidine
3-[(3-hydroxypiperidin-1-yl)methyl]-N-(3-methoxyphenyl)benzamide
N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
methyl 6-(azepan-1-ylmethyl)-3-(2-chloro-6-fluorobenzamido)thieno[2,3-b]pyridine-2-carboxylate
3-{5-[4-(1H-pyrazol-3-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
1-[(5-methylthiophen-2-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
methyl 2-{[(2-chlorophenyl)methyl]sulfamoyl}-6-[(2E)-4-methylpent-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(piperidin-1-ylmethyl)-4-[2-(trifluoromethyl)benzoyl]-1,4-oxazepane
(3-{[(2S,5R)-5-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)oxolan-2-yl]methyl}phenyl)methanamine