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(3S,5R)-N3-cyclopropyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
3-(1-{5-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-cyclopropyl-5-{4-[(pyrimidin-2-yl)amino]piperidine-1-carbonyl}pyrimidin-4-ol
2-methyl-9-(1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(quinoxalin-2-yloxy)hex-5-en-1-yl]piperidine-4-carboxylic acid
(1S,5R)-3-(7-methoxy-4-methylquinolin-2-yl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-hydroxy-2-(pyridin-4-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(3-methylbut-2-en-1-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-cyclopentyl-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-cyclopropyl-1-(2,5-dichlorophenyl)-5-(2-methanesulfonylethyl)-1H-1,2,4-triazole
[(3R,4R)-1-(5-fluoro-2-methylbenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
8-(1,7-dimethyl-1H-indole-2-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3aS,6aS)-5-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-1-oxo-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1R,2S)-N-butyl-2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}cyclohexane-1-carboxamide
2-cyclobutyl-5-fluoro-1-[1-(2,3,4-trimethoxybenzoyl)piperidin-4-yl]-1H-1,3-benzodiazole
5-{[(5-ethyl-2-methylpyrimidin-4-yl)amino]methyl}-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[7-methoxy-2-oxo-4-(piperidin-4-yl)-1,2,3,4-tetrahydroquinolin-6-yl]butanamide
N,N-dimethyl-5-[4-(piperidin-1-yl)butanoyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-(2,6-dichlorophenyl)-1-(thiolan-3-yl)-1H-imidazole
3-{[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}pyridin-2-amine
4-[2-(1-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-2-yl)ethyl]morpholine
5-[(2E)-but-2-en-1-yl]-3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
8-(1,3-benzothiazol-2-ylmethyl)-1-benzyl-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)piperidin-1-yl]ethan-1-one
1,9-dimethyl-4-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(3-methoxypropyl)-8-(4-methoxypyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
6-methyl-3-[(2S)-2-(piperidine-1-carbonyl)pyrrolidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
2-methyl-5-({3-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)-1,3-benzothiazole
3-(2-fluorophenyl)-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)benzamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-oxo-N-propyl-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]-4-methyl-1H-imidazole-2-carboxamide
1-(5-methoxy-2-{[(3-methoxypropyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
2-methyl-1-(2-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-oxoethyl)-1,4-dihydroquinolin-4-one
3-{5-[6-(piperidin-1-yl)pyrimidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-[3-(2H-1,3-benzodioxol-5-yl)-1-methyl-1H-1,2,4-triazol-5-yl]morpholine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(methylamino)-1,3-thiazole-4-carboxamide
3,3-dimethyl-1-({5-[(2-phenylpyrimidin-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
4-{[2-(dimethylamino)ethyl]amino}-N-(2-hydroxybutyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-(4-methylpiperidin-1-yl)-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-(piperidin-3-yl)benzamide
N-[(3S,4R)-1-(3,6-dimethylpyrazin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
6-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1-(1-methyl-1H-indazol-6-yl)urea
2-(4-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-2-methyl-1,3-thiazole-4-carboxamide
(2S,4S)-4-amino-1-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-2-carboxamide
(3S,4S)-1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(piperidin-1-yl)pyrrolidin-3-ol
(1H-indol-2-ylmethyl)({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
(1S,5R)-6-benzyl-3-(6-methylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-({[3-(4-hydroxyphenyl)propyl]carbamoyl}amino)-2-methyl-N-(2-methylpropyl)benzamide