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1-(3-methyl-1,2-oxazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
1-[(2S)-2-(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane-6-carbonyl)pyrrolidin-1-yl]ethan-1-one
N-[(3R,4S)-1-(carbamoylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1,8-dimethyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aS)-2-cyclohexyl-5-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[6-(1H-pyrazol-3-yl)pyrazine-2-carbonyl]morpholine
2-(2-fluoro-6-methoxyphenyl)benzamide
2-(4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
N3-benzyl-N5-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[(3-methoxyphenyl)methyl]-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperazin-2-one
5-methoxy-2-({3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
methyl[3-(4-methyl-1,3-thiazol-5-yl)propyl][(4-methyl-1H-imidazol-2-yl)methyl]amine
1-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2,3,4,9-tetrahydro-1H-carbazole
2-({[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-N-[(2-fluorophenyl)methyl]acetamide
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-1,4-diazepan-2-one
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-8-fluoroquinoline-2-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidine-1-carboxamide
N-methyl-2-[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]-N-(thiophen-3-ylmethyl)acetamide
2-hexanoyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-{[3-(difluoromethoxy)phenyl]methyl}-3-azaspiro[5.5]undecan-9-amine
N-[(2R,4R,6S)-2-cyclohexyl-6-(4-methanesulfonylphenyl)oxan-4-yl]acetamide
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-7-fluoro-2-methylquinoline-4-carboxamide
N-methyl-4-{2-oxa-7-azaspiro[4.5]decane-7-sulfonyl}thiophene-2-carboxamide
2-cyclopropyl-8-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-amino-4-ethyl-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]-1,3-thiazole-5-carboxamide
1-(5-chloro-2-methoxyphenyl)-3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}urea
2-ethyl-1-[(2-methoxyphenyl)methyl]-3-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1,4-dihydropyridin-4-one
[3-(2-methoxyethyl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-3-yl]methanol
N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-2-(pyrrolidin-3-yl)benzamide
5-chloro-3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{2-methylimidazo[1,2-a]pyrimidine-3-amido}-N-phenylpiperidine-1-carboxamide
N-[2-(cyclohexylsulfanyl)ethyl]-3,4-dimethyl-5-sulfamoylbenzamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl]methanol
4-methyl-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1,2,3-thiadiazole-5-carboxamide
1-{5-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
5-{2-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2-aminopyrimidin-4-yl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylic acid
7-(1-benzofuran-2-sulfonyl)-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-(2-methoxyphenyl)-4-[1-(propan-2-yl)piperidin-3-yl]piperazine
4-(4-chlorophenoxy)-N-[1-(3-methylpyridin-2-yl)ethyl]piperidine-4-carboxamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
5-methoxy-3-methyl-2-[4-(thian-4-yl)piperazine-1-carbonyl]-1H-indole
2-ethyl-9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-5-{1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
methyl[2-(phenylsulfanyl)ethyl]{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
N-methyl-N-[(5-methylfuran-2-yl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide