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9-[2-(dimethylamino)acetyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-benzyl-3-ethyl-1-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,4-diazepan-5-one
methyl (2S)-2-[2-(2-phenyl-1,3-thiazol-4-yl)acetamido]propanoate
8-methoxy-4-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
[(3S,5R)-5-[(dimethylamino)methyl]-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]piperidin-3-yl]methanol
2-{2-[6-amino-5-cyano-4-(oxolan-3-yl)pyridin-2-yl]phenoxy}acetamide
2,4-dimethyl-N-[4-(5-methylfuran-2-amido)phenyl]-1,3-oxazole-5-carboxamide
6-methyl-2-{1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
1-(2-methoxyacetyl)-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}piperidine-3-carboxamide
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-3-(3-ethylphenoxy)azetidine
1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(naphthalen-2-ylmethyl)-1,4-diazepan-5-one
1-cyclopropyl-6-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-3-carboxamide
N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N-ethylpyrrolidine-3-carboxamide
1-(4-chlorophenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
7-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-tert-butyl-2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carboxamide
N-[4-(pentyloxy)phenyl]-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
9-(4,5,6,7-tetrahydro-1,3-benzothiazole-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
6-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}pyrimidin-4-ol
N-cyclopentyl-1-[1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
3-cyclopropyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-3-{[(4-methylphenyl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-5-fluoro-1H-indole-2-carboxamide
(1S,5R)-N-(2-chlorophenyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]ethan-1-one
3-(2-{cyclopropyl[(2-ethoxyphenyl)methyl]amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
N-[(3S,4R)-1-[(5-acetylthiophen-3-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
2-(4-{[8-methoxy-2-(4-methoxy-3-methylphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenoxy)ethan-1-ol
1-[cyclohexyl(methyl)amino]-3-(2-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
3-methyl-7-[4-(methylamino)pyrimidin-2-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N,4,6-trimethyl-2-oxo-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-{4-[(2,5-dimethoxyphenyl)methyl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
7-(3-chlorophenyl)-4-(morpholine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3aR,6aS)-5-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[methyl(2-methylpropyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
(1S,2S)-1-phenyl-2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propane-1,3-diol
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-{2-methyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}imidazolidin-2-one
7-methyl-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]-2-fluoro-5-sulfamoylbenzamide
1-[(2-methoxyphenyl)methyl]-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-6-oxopiperidine-3-carboxamide
N-[1-(2-chlorophenyl)ethyl]-1-(4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
2-methoxy-4-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
6-(2,3-difluoro-4-pentylphenyl)-2-methyl-2,3-dihydropyridazin-3-one
1-(4-{3-[({[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}amino)methyl]pyridin-2-yl}piperazin-1-yl)ethan-1-one