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(2S,4R)-4-amino-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-methyl-6-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1H-indole
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
3-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl(quinolin-6-ylmethyl)[(4-{2-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl]amine
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,4-dithiepan-6-amine
2-(4-methoxy-3-methylphenyl)-2-{methyl[2-(pyridin-2-yl)ethyl]amino}acetic acid
N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
N'1-[(3R,4S)-1-(5-chloropyridin-2-yl)-4-propylpyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}pyrimidin-2-amine
1-(3-methylpyridin-4-yl)-4-[(5-methylthiophen-2-yl)methyl]piperazine
N-methyl-4-(piperidin-3-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}benzamide
(1S,5R)-3-[2-(1H-imidazol-1-yl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl[(3-{2-[4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](thiophen-2-ylmethyl)amine
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)furan-3-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[2-(methylsulfanyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
1-(1,2,5-thiadiazole-3-carbonyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
1-[3-(azepane-1-carbonyl)phenyl]-3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]urea
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(quinoxalin-5-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5S)-5-[3-oxo-3-(3-phenoxyazetidin-1-yl)propyl]imidazolidine-2,4-dione
5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrazin-2-ol
N-{1-[1-(3-methylbut-2-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
2-{2-[(3,4-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-N-ethyl-N-methylacetamide
4-[2-(3-fluorophenyl)-1,3-benzoxazole-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,N-dimethyl-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-3-amine
2-amino-4-(3-hydroxyphenyl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
2-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-4-(pyridin-2-yl)pyrimidine
1-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidine
1-[(1R,5R)-3-azabicyclo[3.3.1]nonan-3-yl]-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
8-(2,2-dimethylbutanoyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{[4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-1,2,3,4-tetrazole
N-[4-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)carbamoyl}methoxy)phenyl]propanamide
4-[5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-1,2,4-oxadiazol-3-yl]-1H-indole
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)(2-methylpropyl)amine
2-[4-(1,1-dioxo-1λ6-thiolane-3-carbonyl)piperazin-1-yl]-N-(pyridin-3-yl)acetamide
N-[2-(1H-imidazol-1-yl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-methoxy-4-[4-(2-methoxybenzoyl)piperazin-1-yl]pyridine-3-carbonitrile
(5S)-5-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidin-2-one
2-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
6-(benzyloxy)-4-(furan-3-ylmethyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
3-(3-methylpiperidin-1-yl)-1-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}propan-1-one
3-[(5-ethylpyrimidin-2-yl)amino]-2-(thiophen-2-ylmethyl)propan-1-ol
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-[4-(piperidine-1-carbonyl)morpholin-3-yl]acetamide
N-{[5-(furan-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}methanesulfonamide
3-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(4-fluorobenzoyl)piperidine
4-(propan-2-yl)-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
1-methyl-4-(4-phenyl-1H-imidazole-5-carbonyl)piperazine-2-carboxylic acid
(2S)-1-({2-[3-(1H-imidazol-1-yl)propoxy]-3-methoxyphenyl}methyl)pyrrolidine-2-carboxamide