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2-(4-{[3-(2-phenylethyl)piperidin-1-yl]methyl}phenoxy)acetic acid
2-ethoxy-3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
ethyl({[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[(2-ethylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(ethylamino)pyrimidine-5-carbonyl]piperidin-3-ol
1-[2-(1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
1-methyl-3-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-(quinolin-3-ylmethyl)urea
1-[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(1H-imidazol-2-yl)ethyl]-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
N-{2-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}acetamide
methyl (2S)-2-{[1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-3-yl]formamido}-3-phenylpropanoate
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[3-(pyridin-4-yl)propyl]pyrimidin-2-amine
N-[3-(2-methylpyrimidin-4-yl)phenyl]-2-(pyrrolidin-3-yl)benzamide
5-(dimethylamino)-2-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-2,3-dihydropyridazin-3-one
N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-2-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,3-thiazole-4-carboxamide
N-[3-(3,4,5-trimethoxyphenyl)phenyl]acetamide
1-{2-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
ethyl 4-(2-phenoxyethyl)-1-(thiophene-3-carbonyl)piperidine-4-carboxylate
(2S,4S)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-ethyl-4-[3-(methylsulfanyl)propanamido]pyrrolidine-2-carboxamide
4-[2-(benzenesulfonyl)ethyl]-1-[(2,4-dimethylphenyl)methyl]-1,4-diazepan-5-one
1-[(3S,4R)-1-[2-(2-chlorophenoxy)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-[2-(morpholin-4-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(diethylamino)-3-[4-({[(2,6-dimethoxyphenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
1-(4-acetamido-3-methoxyphenyl)-1H-imidazole-4-carboxylic acid
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]pyrazine-2-carboxamide
3-[(3R,4S)-3-acetamido-4-propylpyrrolidin-1-yl]-N-[(4-fluorophenyl)methyl]propanamide
2-(1-methyl-1H-imidazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(3-chlorophenyl)methyl]-3-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}propanamide
(4aR,7aS)-4-(dimethyl-1,3-oxazole-4-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-{1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
2-({ethyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)benzoic acid
4-[6-(methoxymethyl)pyrimidin-4-yl]-1-methylpiperazine-2-carboxylic acid
(1R,3S)-3-(2-hydroxyethoxy)-7-(2-phenylbenzoyl)-7-azaspiro[3.5]nonan-1-ol
3-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
4-methyl-6-{spiro[azepane-4,2'-chromene]-1-yl}pyrimidin-2-amine
(4aS,7aR)-1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,9S)-11-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylpyridine-3-carboxamide
5-(2-fluorophenoxymethyl)-N-(1-propylpiperidin-4-yl)-1H-pyrazole-3-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-5-methyl-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-[3-(pyridin-2-yl)propanoyl]pyrrolidine-2-carboxamide
2-methyl-6-{[4-(1-phenyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}pyrimidin-4-ol
N-[(1-cyclopentylpiperidin-4-yl)methyl]-4-oxo-N-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
1-cyclopentyl-3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}piperidine
4-[1-(morpholine-4-sulfonyl)piperidin-3-yl]benzoic acid
2,3-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1H-indole-5-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(5S,9aS,9bS)-5-[4-methoxy-3-(methoxymethyl)phenyl]-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one