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methyl 3-[({5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl}formamido)methyl]-5-[2-(thiophen-3-yl)acetamido]benzoate
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]acetamide
7,7-dimethyl-2-(4-propyl-4H-1,2,4-triazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-(benzenesulfonyl)-3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(3R,4R)-4-(azepan-1-yl)-1-[1-(2-chlorophenyl)piperidin-4-yl]piperidin-3-ol
N-{2-[2-(cyclohexylmethyl)morpholin-4-yl]-2-oxoethyl}acetamide
5-chloro-3-methyl-N-[(1s,4s)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexyl]-1H-indole-2-carboxamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-4-(piperidin-1-ylmethyl)benzamide
(4aS,7aR)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{5-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-methyl-1,2-oxazole
N-(2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
N3-tert-butyl-4-oxo-1-(propan-2-yl)-N5-[2-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-{[7-chloro-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-{3-oxo-3-[9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-2-yl]propyl}acetamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(3-fluorophenoxy)ethan-1-one
1-[1'-(quinolin-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-cyclopentyl-N-{[3,5-dimethoxy-4-(oxolan-2-ylmethoxy)phenyl]methyl}thiophene-2-sulfonamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(pyridin-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-{[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]amino}-N-(2-methoxy-5-methylphenyl)acetamide
2,5-dimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(2-hydroxy-3-methylbutanoyl)-N-(5-methyl-1,2-oxazol-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
methyl (2S,4S)-4-(2-hydroxyacetamido)-1-methylpyrrolidine-2-carboxylate
N-[2-(3,4-dimethylphenoxy)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(4aS,7aR)-1-(pyridin-4-ylmethyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 1-(4-tert-butylphenyl)-1H-imidazole-2-carboxylate
2-methyl-6-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}pyridine
2-(4-{1-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)ethan-1-ol
1-({5-[(5-acetylthiophen-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
1-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}-3,5-dimethyl-1H-pyrazole
N-[1-(5-methylpyridin-2-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(morpholin-4-yl)butanamide
(3S,9aR)-3-benzyl-8-(4-fluorobenzoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-cyano-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]pyridine-3-carboxamide
2-(pyrimidin-2-yl)benzonitrile
4-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butan-1-ol
methyl 3-(2-chlorobenzenesulfonamido)-5-[(cyclobutylformamido)methyl]benzoate
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
1-[(2-aminopyridin-3-yl)methyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N,N,3,6-tetramethyl-2-[2-(3-methylbutyl)pyrimidin-5-yl]quinoline-4-carboxamide
2-ethyl-N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}pyrimidine-5-carboxamide
3-benzyl-4-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-2-one
2-(2,4-difluorophenyl)-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
N-(2-chlorophenyl)-3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
(benzylsulfamoyl)[3-(2-chlorophenoxy)propyl]methylamine
1-{2-oxa-7-azaspiro[4.5]decan-7-yl}-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butan-1-one
1-(4-chlorophenyl)-N-(2-{5-[(2,3-dihydroxypropyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)cyclopropane-1-carboxamide
(2S,4R)-N-ethyl-1-(furan-3-ylmethyl)-4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamido]pyrrolidine-2-carboxamide
(1R,2R,4R)-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-ethylbicyclo[2.2.1]hept-5-ene-2-carboxamide
N-methyl-N-{[3-methyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}aniline