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4-(1-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)pyrimidine
1-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
2-(cyclopropylmethyl)-8-(3-hydroxy-4-methoxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-1-{[2-(pyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]sulfonyl}pyrrolidin-3-amine
1-(furan-2-carbonyl)-N-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-amine
1-(cyclohex-3-en-1-ylmethyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-cycloheptyl-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]piperidine-1,3-dicarboxamide
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetamide
N-[4-(3-chloropyridin-4-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]thiophene-2-carboxamide
(1R,2R)-1-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-2,3-dihydro-1H-inden-2-ol
3-{[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl}benzonitrile
1-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
1-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-3-(pyridin-3-yl)propan-1-one
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidin-2-amine
2-[3-(3-hydroxy-3-methylbutyl)benzoyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
1-{2-[7-(2-hydroxyethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-3,3-dimethylurea
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(pyridin-3-yl)ethan-1-one
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-2,4-dimethylpyrimidine
(1S,5R)-6-(cyclobutylmethyl)-3-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1,3-diphenyl-1H-pyrazol-5-yl)-2-(1H-imidazol-1-yl)acetamide
9-[2-(3-fluorophenyl)acetyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-({[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}amino)pyridine-3-carboxylic acid
(3S,4S)-4-cyclopropyl-1-(2-ethylbenzoyl)pyrrolidine-3-carboxylic acid
(3R,4S)-4-{[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](ethyl)amino}oxolan-3-ol
3-{3-[3-(6-methoxypyridin-2-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
(2-methoxyethyl)(methyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
3-(1,3-benzothiazol-2-yl)-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}propan-1-one
4-{5-[(S)-methoxy(phenyl)methyl]-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl}-3-methylpyridine
(1R,3R)-N1-[1-(2,3-dimethylphenyl)piperidin-4-yl]cyclopentane-1,3-diamine
4-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
6-methyl-1-{2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2-dihydropyridin-2-one
1-(furan-2-yl)-2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}ethane-1,2-dione
3-(2-fluorophenyl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-3-phenylpropanamide
4-(4-methoxyphenoxy)-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine
6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purine
1-(3-fluoro-2-methoxybenzoyl)-4-[(3-methylphenyl)methyl]piperazine
(2R,4S)-4-hydroxy-1-[2-(naphthalen-1-yl)acetyl]piperidine-2-carboxylic acid
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-2-(3-hydroxyazetidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-[1-(methoxymethyl)cyclopentyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxylic acid
butyl 2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxylate
5-tert-butyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1,3,4-oxadiazol-2-amine
(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-5-methyl-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-[4-(morpholin-4-ylmethyl)phenyl]-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
1-(4-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}thiophen-2-yl)ethan-1-one
2-[2-(dimethylamino)ethyl]-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
10-methoxy-5-{2-methyl-2,8-diazaspiro[4.5]decane-3-carbonyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide
(4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)methanol