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(1R,4S)-N-ethyl-1,7,7-trimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methylpiperidine-2-carboxamide
ethyl 1-[(2-ethylphenyl)carbamoyl]-4-(2-phenylethyl)piperidine-4-carboxylate
1-{4-[3-({[(2-ethoxyphenyl)methyl]amino}methyl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
2-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
2-{4-[4-(dimethylamino)phenyl]-3,5-dimethyl-1H-pyrazol-1-yl}-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
ethyl 2-[7-(2-methoxybenzoyl)-2,7-diazaspiro[4.5]decan-2-yl]acetate
4-{[(1-methylazepan-2-yl)formamido]methyl}benzoic acid
N-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
(3R,4R)-4-(azepan-1-yl)-1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-ol
N-(2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}ethyl)acetamide
4-chloro-1-methyl-3-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}-1H-indazole
2-(1H-1,3-benzodiazol-1-yl)-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpropanamide
N2,N2-dimethyl-6-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,3,5-triazine-2,4-diamine
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-methoxyethan-1-one
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(carbamoylmethyl)propanamide
3-(azepane-1-carbonyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[5-(4-cyclohexylphenyl)-1,2,4-triazin-3-yl]-N,N-dimethylpyrrolidin-3-amine
2-(1-ethyl-1H-pyrazol-4-yl)-3,6-dimethyl-4-(2-methylpiperidine-1-carbonyl)quinoline
6-methyl-2-(pyridin-3-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]pyrimidin-4-amine
7-methyl-2-(morpholine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(4aS,8aS)-2-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-decahydroisoquinolin-4a-ol
3-{2-oxo-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]ethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2-(pyridin-4-ylsulfanyl)acetamide
5-(propan-2-yl)-3-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}pyrrolidin-2-yl)-1,2-oxazole
4-[4-(3-methylpiperidine-1-carbonyl)piperidin-1-yl]-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
[(2S,4R)-4-(dimethylamino)-1-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-2-yl]methanol
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
[(4aS,8aR)-6-(1,7-dimethyl-1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
N-[2-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-2-carboxamide
2-[(1-methyl-1H-indol-6-yl)methyl]-2-azaspiro[4.4]nonane
1-(azepan-1-yl)-3-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-2-methoxyphenoxy}propan-2-ol
1-(benzenesulfonyl)-4-[(2-butyl-1H-imidazol-4-yl)methyl]piperazine
2-methyl-1-{7-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}butan-1-one
4-methyl-2-{2-[(3-propyl-1H-pyrazol-5-yl)formamido]ethyl}-1,3-thiazole-5-carboxylic acid
N-methyl-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(oxan-4-ylmethyl)piperidine-4-carboxamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[3-(dimethylamino)propyl]-N-methylpyrimidin-2-amine
4-[(2-methylprop-2-en-1-yl)oxy]-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}benzamide
6-tert-butyl-N,1-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(dimethylamino)-1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethan-1-one
4-ethyl-1-[(5-fluoro-2-methylphenyl)methyl]-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,5R)-5-(morpholine-4-carbonyl)-N-(quinolin-2-ylmethyl)piperidine-3-carboxamide
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(4-methoxy-3-methylphenyl)methyl]piperidine
4-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
4-[4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
5-methyl-4-{[1-(1H-1,2,4-triazol-5-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
1-methyl-4-[4-(trifluoromethyl)pyridin-2-yl]piperazine-2-carboxylic acid