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1-amino-N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)cyclopropane-1-carboxamide
6-[({[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amino)methyl]-1,4-oxazepan-6-ol
4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline
(1R,7S)-6-(3-hydroxyazetidine-1-carbonyl)-3-[(3-methoxyphenyl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1'-[(2-fluorophenyl)methyl]-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-(2-phenylethyl)-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decane
3-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)-1-(4-methylphenyl)urea
4-({1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}methyl)morpholine
(3S,4R)-1-(4-chloro-2-methoxybenzoyl)-4-methylpiperidine-3,4-diol
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
methyl 3-[(2,2-dimethylpropanamido)methyl]-5-(furan-2-amido)benzoate
5-[(1-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one
(1S,5R)-3-(2-aminopyrimidin-4-yl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
[1-(quinolin-4-ylmethyl)azepan-2-yl]methanol
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
5-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]isoquinoline
5-chloro-6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxylic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(4-methylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[3-(morpholin-4-ylmethyl)phenyl]-1,2-dihydropyridin-2-one
3-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
4-(3-fluorophenoxy)-1-(quinolin-2-yl)piperidine-4-carboxylic acid
N-cycloheptyl-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-cyclobutyl-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
5-[2-(benzenesulfonyl)ethyl]-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazole
6-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-methyl-1-benzofuran-5-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]acetamide
4-{4-[1-(2,3-dihydro-1H-inden-5-yl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
methyl[1-(4-methylpyridin-2-yl)propan-2-yl][(3-methylthiophen-2-yl)methyl]amine
1-(2-{2-[2-(propylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)imidazolidin-2-one
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
4-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
1-(oxan-4-yl)-3-[2-(pyridin-2-ylmethoxy)phenyl]urea
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
4-methoxy-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
2-{1-[(4-ethoxyphenyl)methyl]-4-(thian-4-yl)piperazin-2-yl}ethan-1-ol
6-({[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}propanamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[3-(pyridin-2-yl)propyl]acetamide
1-cyclopentyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
2-(3-chloro-4-hydroxyphenyl)-1-[(3S)-3-ethylmorpholin-4-yl]ethan-1-one
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(5-methylfuran-2-yl)methyl]acetamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
2-cyclobutyl-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-5-(2-methoxyacetamido)-N,1-dimethyl-1H-1,3-benzodiazole-7-carboxamide
5-methyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
8-[4-(4-chlorophenyl)butanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{2,7-diazaspiro[4.5]decane-7-carbonyl}-2-methyl-N-(pyridin-3-ylmethyl)aniline