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1-methyl-4-[(3-methylpyridin-4-yl)methyl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
(3R,4R)-3,4-dimethyl-1-(4-propylpyrimidine-5-carbonyl)pyrrolidin-3-ol
N-methyl-3-{[4-(2-methyl-5-propylpyrimidin-4-yl)piperazin-1-yl]methyl}pyridin-2-amine
1-[3-(1H-imidazol-2-yl)benzoyl]azocane
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(3-chloro-5-fluorophenyl)pyridine-3-carbonitrile
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(3-hydroxypropanoyl)piperidine-4-carboxamide
3-(but-2-yn-1-yl)-5-[1-(1H-imidazole-4-carbonyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
[(5-chloro-2,3-dimethoxyphenyl)methyl](methyl)(oxan-4-ylmethyl)amine
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-(5-acetylthiophen-3-yl)-1-{2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}ethan-1-one
(3S,5R)-1-[(3-methoxyphenyl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-(3-fluorophenyl)-5-(1H-imidazol-2-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
1'-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(2-methoxyethyl)-9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{[3-(2-aminoethyl)phenyl]methyl}-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
4-(4-chlorophenoxy)-1-(pyrazin-2-yl)piperidine-4-carboxylic acid
4-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}benzoic acid
6-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]isoquinolin-3-amine
(2S,4R)-4-benzamido-N-ethyl-1-[2-(1H-imidazol-1-yl)acetyl]pyrrolidine-2-carboxamide
N-[(4-methoxyphenyl)methyl]-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
8-methoxy-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
1-(2-methoxy-4-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
4-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N,N-dimethylaniline
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
N-[4-(methylamino)butyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
4-[2-(2-ethylphenoxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
3-[ethyl(methyl)amino]-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
3-(3-methoxyphenoxymethyl)-1-(oxane-4-carbonyl)piperidine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(1H-1,2,4-triazol-1-yl)acetamide
N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-4-phenylazepane
(1S,2S,9S)-11-{2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetyl}-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
6-methyl-5-[5-(2-methylprop-1-en-1-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
1-[(4-fluoro-3-methoxyphenyl)methyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-phenylpiperidine-4-carbonitrile
(3R,4R)-4-ethyl-1-{5-[(phenylsulfanyl)methyl]furan-2-carbonyl}piperidine-3,4-diol
5-[1-butyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]-2,2-dimethylthiomorpholin-3-one
2-[4-(1H-indol-5-yl)-6-methylpyrimidin-2-yl]phenol
1-(cyclopentylmethyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(2S,4R)-4-amino-N,N-diethyl-1-(4-propoxybenzoyl)pyrrolidine-2-carboxamide
N-(2-chlorophenyl)-3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}propanamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methoxyethan-1-one
N-(2-hydroxyethyl)-4-({1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}amino)pyridine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
7-[(4-fluorophenyl)methyl]-2-[3-(1H-pyrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2-{[(6-methoxypyrimidin-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-4-({2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-1,3-oxazole
2-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-5-methoxypyridin-4-ol