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methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
N-methyl-2-[methyl(pyridin-3-ylmethyl)amino]-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
(3R,7S,8aS)-7-[({3-[2-(dimethylamino)ethoxy]phenyl}methyl)amino]-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]-1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
4-{[1-(cyclohexylmethyl)-5-(pyrrolidin-3-yl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
3-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
2-[4-(5-{[(2-methoxyphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]propanamide
2-[3-(4-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-[2-(2-methoxyphenyl)ethyl]acetamide
{1-[1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}(methyl)(pyridin-4-ylmethyl)amine
N-{2-[2-(3,5-dimethyl-1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}-N-methylmethanesulfonamide
3-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
ethyl 4-[(4-chlorophenyl)methyl]-1-[1-(4-methylpyridin-2-yl)propan-2-yl]piperidine-4-carboxylate
1-{1-[(2,6-difluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
4-(dimethyl-1,3-thiazole-4-carbonyl)thiomorpholine
3-({2-[2-(ethylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole-5-carboxamide
5-fluoro-2-{1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
3-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
9-(2,3-dihydro-1H-indene-1-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
4-(1H-imidazol-2-yl)-1-{1-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-1H-1,2,3-triazole
2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-6-methylquinolin-4-ol
6-cyclopentyl-1-methyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[2-(1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
5-methyl-4-phenyl-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H-imidazole
(1S,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[1-(thiophen-3-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-methyl-3-[1-(propan-2-yl)-5-[(propan-2-yl)sulfamoyl]-1H-1,3-benzodiazol-2-yl]propanamide
methyl 3-{[1-(cyclopropylmethyl)-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
(1s,4s)-4-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}cyclohexan-1-amine
4-hydroxy-1-[4-(2-methylpropyl)benzoyl]piperidine-4-carboxylic acid
[(3-chloro-4-methoxyphenyl)methyl][(5-cyclopropyl-1H-pyrazol-3-yl)methyl]methylamine
({1-[2-(2-fluorophenoxy)ethyl]-1H-indol-3-yl}methyl)[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]amine
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2,5,7,8-tetramethyl-3,4-dihydro-2H-1-benzopyran-6-ol
(3aR,6aR)-2-acetyl-5-(4-chlorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(4-fluorophenoxy)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(4-methoxypiperidin-1-yl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[2-(2,2-dimethylpropanamido)ethyl]-N-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-{[(3S,4S)-3-hydroxy-1-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl]methyl}pyrrolidine-1-carboxamide
5-methoxy-2-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-N-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-(4-fluoro-3-methylphenyl)-3-[(1-propyl-1H-pyrazol-4-yl)methyl]urea
3-(1H-1,3-benzodiazol-2-yl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
2-(4,5-dimethyl-1H-imidazol-1-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
(1R,5R)-N,N-dimethyl-6-(3-phenylpropanoyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-[4-(adamantan-1-yl)piperazin-1-yl]-3-(1H-imidazol-1-yl)butan-1-one
1-(2,2-dimethylpropyl)-3-hydroxy-3-[(4-phenylpiperazin-1-yl)methyl]piperidin-2-one