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1-(4-cyano-2-ethylphenyl)-3-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]urea
4-methyl-1-{4-oxo-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-6-yl}piperidine-4-carbonitrile
1-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)urea
8-[6-(dimethylcarbamoyl)pyridin-2-yl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[(dimethylamino)methyl]-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)azepan-4-ol
5-methyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,3-benzodiazole-2-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-cyclohexyl-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-(4-{[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]methyl}phenyl)acetamide
2-(dimethylamino)-N-[1-(hydroxymethyl)cycloheptyl]-2-(3-methylphenyl)acetamide
(3-ethyl-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-yl)methanol
2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
N'1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N'1-methylcyclopropane-1,1-dicarboxamide
3-[3-(1H-pyrazol-3-yl)phenyl]phenol
1-(5-methoxyfuran-2-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
6-(4-ethylphenyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-ethyl-2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)-3-propylurea
1-(3-chloro-4-methoxyphenyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
(4aS,7aR)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-3,5-dimethyl-N-(oxolan-2-ylmethyl)furan-2-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
methyl({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})[1-(pyridin-2-yl)propyl]amine
N-{1-[(2-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}morpholine-4-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(oxan-4-yl)-2,8-diazaspiro[4.5]decan-3-one
2-ethyl-N-(1-methanesulfonylpiperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
8-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-cyclopentyl-4-{3-[(pyridin-2-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
8-cyclopropanecarbonyl-2-(6-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 4-{[(2S,4R)-2-({imidazo[1,2-a]pyridin-2-ylmethyl}carbamoyl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidin-1-yl]methyl}benzoate
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3-methoxyphenyl)methyl]acetamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[3-(methylsulfanyl)propyl]piperidine
[(3-chloro-5-fluorophenyl)methyl][(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]methylamine
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]propanamide
5-amino-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-ethyl-1-(3-methoxypropyl)-1H-1,3-benzodiazole-7-carboxamide
6-methyl-3-[2-(4-methylpiperazin-1-yl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-[1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-1-oxopropan-2-yl]pyrrolidin-2-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(propan-2-yloxy)propyl]acetamide
2-(dimethylamino)-4-methyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}pyrimidine-5-carboxamide
2-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-2-yl)pyridine
9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-(5-methylthiophen-2-yl)-4-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(4-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenyl)acetamide
2-(3-chlorophenyl)-1-[1-(hydroxymethyl)-9-propyl-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
N-[(3S,4R)-1-[(2,6-dichloro-3-hydroxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylpyrimidin-2-amine
N-(5-methyl-2-pentanamidophenyl)-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
2-(3-methoxypropyl)-1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidine
1-[4-(pyridin-2-yl)piperazin-1-yl]-3-[1-(quinolin-2-ylmethyl)piperidin-3-yl]propan-1-one
N-(isoquinolin-5-ylmethyl)-N-methyl-4-(1H-pyrazol-3-yl)benzamide
2-{2-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide