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7-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(2R)-2-methoxy-2-phenyl-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-[methyl(pyridin-3-ylmethyl)amino]-1-[4-(4-methylphenoxy)piperidin-1-yl]ethan-1-one
N-[(2-chloro-6-fluorophenyl)methyl]-N,6-diethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
5-[3-({[4-(butan-2-yloxy)-3-methoxyphenyl]methyl}amino)propyl]-1,3,4-thiadiazol-2-amine
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
3-(1H-pyrazol-1-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]benzamide
(2S,4R)-N-ethyl-4-(2-hydroxyacetamido)-1-[(6-methylquinolin-5-yl)methyl]pyrrolidine-2-carboxamide
ethyl 4-(cyclopropylmethyl)-1-[1-(pyridin-3-yl)propan-2-yl]piperidine-4-carboxylate
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
2-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-3-methoxypyrazine
(2R)-2-amino-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N,4-dimethylpentanamide
N-methyl-2-(morpholin-3-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
5-methyl-1-{2-[1-(2-methylphenyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
N-ethyl-4,5-dimethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]thiophene-2-carboxamide
5-chloro-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(methylamino)benzamide
1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethan-1-one
7-cyclohexyl-2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(1R,5R)-6-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{[4-methyl-5-(1-pentylpiperidin-3-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
{3-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]phenyl}methanol
[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl){[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
3-ethyl-6-[4-(pyridin-4-yl)piperazine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
1-methyl-3-(2-methylpropyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(4-chloro-3-fluorobenzoyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-[(oxan-4-ylmethyl)amino]pyridine-3-carboxamide
({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)[(4-methyl-1,3-benzoxazol-2-yl)methyl]amine
3-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
[(2S,4R)-4-(dimethylamino)-1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}pyrrolidin-2-yl]methanol
3-tert-butyl-1-methyl-4-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(4aS,7aR)-1-(1H-imidazol-4-ylmethyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-4-{1,4-dioxa-8-azaspiro[4.5]decan-8-yl}-1-(4-methoxybenzoyl)pyrrolidin-3-ol
2-methyl-5-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}pyridine
methyl 2-(3-methylphenyl)-2-[(2-oxo-1,2-dihydroquinolin-4-yl)formamido]acetate
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1-(4-phenylpiperazin-1-yl)propan-1-one
3-(4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)propan-1-ol
3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-[2-(methylsulfamoyl)phenyl]urea
3-(1H-1,3-benzodiazol-1-yl)-1-[3-(4-fluorophenyl)pyrrolidin-1-yl]propan-1-one
4-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
1-ethyl-N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-[2-(diethylamino)ethyl]-5-(furan-2-yl)-1H-pyrazole-4-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
4-[4-({3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}methyl)phenyl]but-3-yn-1-ol
4-[2-(dimethyl-1,3-thiazol-5-yl)acetamido]-N-phenylpiperidine-1-carboxamide
3-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-[4-(4-methylphenyl)phenyl]urea
5-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
6-{4-[3-(morpholine-4-carbonyl)phenoxy]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one