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methyl 2-[({[2-(morpholin-4-yl)pyridin-3-yl]methyl}carbamoyl)amino]benzoate
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}acetamide
N-[(1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidin-3-yl)methyl]-1H-indole-2-carboxamide
1-(4-fluorophenyl)-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}pyrrolidine
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-(2-methylpropyl)piperidin-4-amine
N-(1-ethyl-1H-pyrazol-5-yl)-2-[4-methyl-3-(1-methyl-1H-pyrazol-5-yl)-1H-pyrazol-1-yl]acetamide
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(pyrrolidine-1-carbonyl)piperidine
ethyl 1-(1-methyl-1H-pyrazole-5-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
2-[2-(pyridin-2-yl)ethyl]-9-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-3-(3-phenylpiperidine-1-carbonyl)-1,2-dihydropyridin-2-one
11-(2H-1,3-benzodioxol-4-yl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
(4aS,8aR)-1-(3-methoxypropyl)-6-(quinolin-4-yl)-decahydro-1,6-naphthyridin-2-one
4-({4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]furan-2-yl}methyl)morpholine
N-methyl-2-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]acetamide
(3S,4R)-3-methoxy-1-(4-methylnaphthalene-1-carbonyl)piperidin-4-amine
2-(2H-1,3-benzodioxole-5-carbonyl)-1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
(1S,6R)-3-{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
1-[(2-fluorophenyl)methyl]-N-[2-(5-methylthiophen-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
5-methyl-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzoxazole
(1R,7S)-3-(2-methoxyethyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-3-(5-methyl-1,2,4-oxadiazol-3-yl)benzamide
9-[3-(morpholin-4-ylmethyl)piperidin-1-yl]-3-azaspiro[5.5]undecane
N-cyclopentyl-2-(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)butanamide
1-[3-(1H-imidazol-2-yl)benzoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,5,7-trimethylpyrido[2,3-d]pyrimidin-4-amine
1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(propan-2-yl)piperazine
N-(1-hydroxy-2-methylpropan-2-yl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
1-(4-{[3-(dimethylamino)propyl](methyl)amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-{2-hydroxy-3-[2-methoxy-4-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
(2E)-N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-3-(pyridin-2-yl)prop-2-enamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]propan-1-one
N-(3-cyano-4-ethoxyphenyl)-3-phenylpiperazine-1-carboxamide
2-(cyclopropylmethyl)-9-[(3R)-3-hydroxy-3-phenylpropyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2,4-dimethoxyphenyl)-3-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}propanamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetamide
(1R,5R)-N,N-dimethyl-6-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(azepane-1-sulfonyl)-5-(1H-pyrazol-4-yl)benzoic acid
8-(2,2-diphenylacetyl)-2,8-diazaspiro[4.5]decan-3-one
1,3-dimethyl-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(1R,3S,5S)-3-(4-methoxyphenyl)-8-{pyrazolo[1,5-a]pyridine-3-carbonyl}-8-azabicyclo[3.2.1]octane
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-{[1-(ethoxymethyl)cyclobutyl]methyl}-1-[4-(methylsulfanyl)phenyl]urea
3-({1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}methyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(5-fluoropyridin-3-yl)-3-[(1,2-oxazol-5-ylmethyl)sulfamoyl]benzamide
N-[2-(2,4-difluorophenyl)-1-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}ethyl]-N-methylpyridine-3-carboxamide
3-(1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-hydroxyethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-2-(pyridin-4-yl)quinoline
7-(3-chlorophenyl)-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-benzyl-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one