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2-{3-[2-(6-methylpyridin-2-yl)-1H-imidazol-1-yl]phenyl}acetic acid
[1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-3-(hydroxymethyl)piperidin-3-yl]methanol
2-cyclopropanecarbonyl-8-[(3,5-dimethylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-[2-(2-hydroxyphenyl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-fluoro-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-benzofuran-2-carboxamide
3-(2-{[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]amino}propyl)-3,4-dihydroquinazolin-4-one
3-methyl-2-{3-methyl-5-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-1,2,4-triazol-1-yl}pyridine
2-methyl-5-{3-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidine-1-carbonyl}-2,3-dihydro-1H-isoindole-1,3-dione
2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-5-fluoro-N-methylpyrimidin-4-amine
N-benzyl-4-oxo-5-(3-phenylpiperidine-1-carbonyl)-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
(1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methanol
2-{1-cyclohexyl-5-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}acetamide
6-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-N-[(1-hydroxycyclohexyl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(1S,5R)-3-benzyl-6-[5-(methoxymethyl)thiophene-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(2R,3R)-3-amino-1'-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
1-benzyl-4-oxo-N3-[(1-phenylcyclohexyl)methyl]-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-fluoro-2-{[3-(3-methoxypropyl)piperidin-1-yl]methyl}-1-methyl-1H-indole
3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-[3-(1,3-oxazol-5-yl)phenyl]piperidine-1-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-(1H-imidazol-1-ylmethyl)cyclopropane-1-carboxamide
4-(2-methylpyridin-4-yl)-N-(1,3,4-thiadiazol-2-yl)-1,4-diazepane-1-carboxamide
4-[(4-methylphenyl)methyl]-3-{2-oxo-2-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethyl}piperazin-2-one
2-[2-(6-methoxypyridin-3-yl)phenyl]ethan-1-amine
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-oxo-1,3-oxazolidine-4-carboxamide
2-{1-[(3-chlorophenyl)methyl]-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-methyl-1H-imidazole
(4aS,7aR)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-chlorophenyl)-3-(2-hydroxyphenyl)-N-(2,2,2-trifluoroethyl)propanamide
4-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyrimidine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-[3-(2-{4-[1-(dimethylamino)ethyl]phenyl}-1H-imidazol-1-yl)phenyl]acetamide
3-cyclopropyl-5-[(oxolan-2-ylmethoxy)methyl]-1-phenyl-1H-1,2,4-triazole
{3-ethyl-1-[1-(3-methoxyphenyl)piperidin-4-yl]piperidin-3-yl}methanol
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(2-methylbutan-2-yl)carbamoyl]pyrrolidine-2-carboxylic acid
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-[3-(2-oxopyrrolidin-1-yl)benzoyl]-1,4-diazepan-2-one
5-(6-methylpyridine-3-carbonyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-({1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}oxy)pyrimidine
2-{4-[(3-chloro-4,5-dimethoxyphenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-[4-(3-fluorophenyl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-2-(ethoxymethyl)pyrrolidine
N-{2-[1-(3-chlorobenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
4-(2-fluorobenzoyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]morpholine-2-carboxamide
N-[(4-phenyloxan-4-yl)methyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3,6,7-trimethyl-N-(pyridin-3-ylmethyl)-1-benzofuran-2-carboxamide
N-(2-methoxyethyl)-1,6-dimethyl-2-oxo-N-(pyridin-4-ylmethyl)-1,2-dihydropyridine-3-carboxamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[3-(prop-2-en-1-yloxy)benzoyl]piperidine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethan-1-one
2-(1H-1,3-benzodiazol-1-yl)-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}acetamide
2-amino-6-(3,5-difluorophenyl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
2-(methylamino)-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}benzoic acid