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N-(4-fluorophenyl)-1-(1-methyl-1,2,3,4-tetrahydroquinoline-6-carbonyl)piperidin-3-amine
N-(1-phenylethyl)-2-(1H-pyrazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(4-fluoro-2-methylbenzoyl)pyrrolidin-3-yl]methanol
2-amino-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-6-hydroxy-5H-indeno[1,2-b]pyridine-3-carbonitrile
(1R,2R,6S,7S)-4-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
(3aR,6aR)-2-methanesulfonyl-5-(quinolin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2,4-dimethoxyphenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
1-[1-(3-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
2-(cyclopropylmethyl)-8-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
(2-{2-[1-(4-chlorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1-tert-butyl-4-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]pyrrolidin-2-one
2-phenyl-N-(pyridin-4-ylmethyl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-methyl-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-(4-fluorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-oxobutanamide
1-[2-(1H-imidazol-2-yl)benzoyl]-3-[(methylsulfanyl)methyl]piperidine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-[4-(3,7-dimethyl-1H-indol-2-yl)-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
N-cyclopropyl-1-[2-(piperidin-2-yl)ethyl]-N-(thiophen-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
1-(3,4-dimethylphenyl)-N-(1H-indol-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-{1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidine-4-carbonyl}piperidin-3-ol
N-[3-(1,3-benzothiazol-2-yl)propyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-(2-hydroxy-3-phenoxypropyl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
3-[1-(1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)piperidin-3-yl]benzoic acid
4-[1-(benzenesulfonyl)cyclopropanecarbonyl]-2-(trifluoromethyl)morpholine
4-{6-[1-(6-methoxypyrimidin-4-yl)piperidin-3-yl]-2-methylpyrimidin-4-yl}morpholine
(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-propylpiperidin-3-yl)methanol
1-(2-phenylethyl)-4-(1H-pyrazol-3-ylmethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
1-[(5-cyclopentylthiophen-2-yl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
3-(3-methoxypiperidine-1-carbonyl)-N-(1H-pyrazol-3-ylmethyl)benzene-1-sulfonamide
N-(2-{7-[(3-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
N-(furan-2-ylmethyl)-1-methyl-N-(3-methylbutan-2-yl)-5-oxo-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-methyl-5-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl]-2-oxo-1,2-dihydropyridine-3-carbonitrile
6-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]pyridine-3-carboxylic acid
(1R,3S)-7-[4-(trifluoromethyl)benzoyl]-7-azaspiro[3.5]nonane-1,3-diol
4-[2-(cyclohexylmethyl)morpholine-4-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
2-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-{1-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]piperidin-3-yl}-3-phenylpropan-1-one
1,3-dimethyl-N-[3-(methylsulfanyl)propyl]-1H-indole-2-carboxamide
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-(1H-indol-3-yl)propan-1-one
ethyl(furan-3-ylmethyl)({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amine
2-[(3-methoxyphenyl)amino]-N-[4-(pyrrolidin-1-yl)butyl]butanamide
4-{4-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pyrimidin-2-amine
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-1-(3-{5-methyl-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)ethan-1-one
(1S,5R)-6-(cyclobutylmethyl)-3-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[3-(difluoromethoxy)phenyl]-3-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}urea
N,N-diethyl-2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]acetamide
7-(5-chloropyridin-2-yl)-4-(2-hydroxypropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl[(3-methylquinoxalin-2-yl)methyl](1,3-thiazol-2-ylmethyl)amine
5-methyl-N-{[3-methyl-7-(3-phenylprop-2-ynoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-carboxamide