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4,4,4-trifluoro-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)butanamide
5-cyclopropyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
N-({4-hydroxy-1-[2-(1H-imidazol-1-yl)acetyl]azepan-4-yl}methyl)morpholine-4-carboxamide
N-methyl-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
2-(3-oxopiperazin-1-yl)-2-(thianthren-1-yl)acetic acid
2-[(4-benzylpiperazin-1-yl)methyl]-N-(furan-2-ylmethyl)-N-methyl-1,3-oxazole-4-carboxamide
(1H-imidazol-4-ylmethyl)(methyl)[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]amine
N-[1-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopentanecarboxamide
2,3-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-(1-carbamoylcyclopentyl)-7-chloro-2-methylquinoline-4-carboxamide
3-{[4-(2-methyl-5-propylpyrimidin-4-yl)piperazin-1-yl]methyl}-4H-chromen-4-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl})amine
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}piperidine-3-carboxamide
3-(oxolan-3-yl)-5-[2-(pyrrolidin-1-yl)phenyl]-1,2,4-oxadiazole
7-(pyridin-3-ylmethyl)-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methoxybenzamide
1-(furan-2-yl)-2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethane-1,2-dione
3-(2,5-dimethoxyphenyl)-1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidine
{5-[1-(1H-indol-2-ylmethyl)-1H-imidazol-2-yl]furan-2-yl}methanol
dimethyl(2-{2-[1-(pyridine-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
4-[(3aR,6aR)-2-acetyl-octahydropyrrolo[3,4-c]pyrrole-3a-amido]-N-ethylpiperidine-1-carboxamide
(3S,4S)-1-[5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carbonyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
N-ethyl-5-[4-(2-methoxyphenyl)piperidine-1-carbonyl]pyrimidin-2-amine
methyl 3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-4-ylmethyl)piperidin-3-yl]propanoate
dimethyl({2-[2-methyl-5-(propan-2-yl)pyrimidin-4-yl]phenyl}methyl)amine
N-[(4-fluorophenyl)methyl]-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-(prop-2-en-1-yl)butanamide
N-ethyl-2,2-dimethyl-N-[(2-methyl-1H-imidazol-4-yl)methyl]oxan-4-amine
N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]thiophene-2-carboxamide
5-methyl-2-(3-methylthiophen-2-yl)-4-{1H-pyrazolo[3,4-b]pyridin-1-ylmethyl}-1,3-oxazole
4-benzyl-1-[(4-fluorophenyl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(3,4-difluorophenoxymethyl)-N-methyl-N-[3-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
4-methyl-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)pyridine-3-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)pyrrolidin-3-yl]acetamide
3-[5-(3,4-difluorobenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1,9-dimethyl-4-[(3E)-pent-3-enoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{4-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
1-ethyl-5-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
1-(3-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}propyl)piperidin-3-ol
2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[(2S)-2-hydroxypropyl]acetamide
3-(4-methyl-1,3-thiazol-5-yl)-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
1-cyclopentyl-4-oxo-N3-(propan-2-yl)-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-3-methylbut-2-en-1-one
ethyl 1-[(2E)-2-methylbut-2-en-1-yl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
3-(3-methoxyphenyl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
2-methyl-4-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}phenyl)butan-2-ol
1-{1-[(4-ethylphenyl)methyl]-1H-1,2,4-triazol-5-yl}-3-(methylsulfanyl)propan-1-ol
(4aS,8aR)-6-(2-aminoacetyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one