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methyl 2-[(4-fluorophenyl)sulfamoyl]-6-(3-methylbenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
6-(aminomethyl)-N-(1H-imidazol-2-ylmethyl)-N,2-dimethylpyrimidin-4-amine
9-(2-ethoxypropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-3-phenyl-N-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)-N-(3-methoxyphenyl)piperidine-1-carboxamide
1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
{4-[6-(trifluoromethyl)pyridin-2-yl]phenyl}methanol
3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-one
1-{2-[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]pyrimidin-4-yl}piperidin-3-ol
3-{[1-(4-fluorobenzenesulfonyl)pyrrolidin-3-yl]methyl}benzamide
3-(4-methyl-2-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)-1,3-oxazolidin-2-one
3-{5-[3-(2-methyl-1H-indol-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-[3-(dimethylamino)propyl]-8-(thiophen-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,7S)-5-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-(dimethyl-1,2-oxazol-4-yl)-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidin-4-amine
1-(1H-imidazol-4-ylmethyl)-4-(4-methoxyphenyl)-2-methylpiperazine
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
N-(3,4-dimethoxyphenyl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
(1S,5R)-3-benzyl-6-[4-(methylsulfanyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-amino-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pent-2-yn-1-yl)pyrrolidin-3-yl]-4-methyl-1,3-thiazole-5-carboxamide
6-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
2-amino-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4-methyl-1,3-benzothiazole-6-carboxamide
N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
2-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}pyridine
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(1-ethyl-1H-pyrazol-3-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-indol-3-yl)propan-1-one
N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
6-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]hexan-1-ol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-1-(2-phenylphenyl)piperazin-2-one
N-[1-(2,4-dimethylphenyl)ethyl]-N'-(2-methylphenyl)propanediamide
N-[1-(1-{[3-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
6-[1-cyclohexyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N-(4-carbamoyl-3-chlorophenyl)-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
N-(1,2-diphenylethyl)-2-ethyl-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1'-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-(furan-2-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(2S,4S)-4-amino-1-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
5-({[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-4-(oxolan-2-ylmethyl)piperazine
5-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}-2-phenyl-1,3-thiazole
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-chlorobenzamide
(3S,9aR)-3-(cyclohexylmethyl)-8-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2,2-dimethyl-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}methyl)propanamide
4-(hydroxymethyl)-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
5-methyl-N-[4-(morpholin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,2-oxazole-4-carboxamide