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(1S,5R)-6-[4-(methylsulfanyl)benzoyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-cyclohexyl-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
methyl (2S)-1-{2-[benzyl(methyl)amino]-6-phenylpyridine-3-carbonyl}pyrrolidine-2-carboxylate
(1S,5R)-3-(6-methylpyridazin-3-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(1H-imidazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
2-(2-{[2-(dimethylamino)-6-ethylpyrimidin-4-yl]amino}ethyl)-1,2-dihydrophthalazin-1-one
3-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-1-(2-chloro-5-methylphenyl)-3-methylurea
ethyl 5-{[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]methyl}furan-2-carboxylate
1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
methyl 1-{2-hydroxy-3-[4-({[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-2,6-dimethylpyridine-4-carboxamide
7-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-1H-indole
methyl 4-({3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}methyl)benzoate
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(2-phenylethyl)piperidine-4-carboxamide
2-{4-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}amino)methyl]phenoxy}ethan-1-ol
1-[(2-fluorophenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
4-benzyl-1-[(dimethyl-1,3-thiazol-2-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-cyclopropyl-N-ethyl-6-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-1,6-dihydropyrimidine-5-carboxamide
methyl(2-methylpropyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
2-amino-N-methyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-benzothiazole-5-carboxamide
8-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-2,6-dimethyloctan-2-ol
1-(dimethylamino)-3-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)propan-2-ol
3-(1H-imidazol-4-ylmethyl)-4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperazin-2-one
8-(1,3-benzoxazol-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-(6-methylpyridin-2-yl)piperazine
2-amino-8-{2-[3-(1H-imidazol-1-yl)propoxy]phenyl}-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
N-[2-(4-methoxyphenyl)ethyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4S)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
4-cyclobutyl-2-(4-methanesulfonylphenyl)-6-methylpyrimidine
8-[4-(1H-pyrazol-1-yl)benzenesulfonyl]-2,8-diazaspiro[4.5]decan-3-one
4-[2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)ethyl]benzene-1-sulfonamide
1-(1-benzylpyrrolidin-3-yl)-4-(1-propyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
3-(3-chloro-1,2-oxazol-5-yl)-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]propan-1-one
1-methyl-1-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
1-methyl-3-phenyl-8-(thiophen-3-ylmethyl)-1,8-diazaspiro[4.5]decan-2-one
2-(3-fluorophenoxymethyl)-N-(2,2,2-trifluoroethyl)-1,3-oxazole-4-carboxamide
(1R,5R)-3-methanesulfonyl-6-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-[2-(1H-imidazol-4-yl)ethyl]-9-(2-phenylpropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-fluoro-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N,6-dimethylimidazo[1,2-a]pyridine-2-carboxamide
2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-N-[(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)methyl]acetamide
N-[(2-chlorophenyl)methyl]-2-cyclopropyl-N-(2-methoxyethyl)-6-oxo-1,6-dihydropyrimidine-5-carboxamide
1-cyclobutanecarbonyl-4-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]piperidine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-[(dimethylcarbamoyl)amino]-N-methylacetamide
3-{5-[(5-propylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
1-{[(3R,4R)-4-(hydroxymethyl)-1-[(2-methoxy-3,5-dimethylphenyl)methyl]pyrrolidin-3-yl]methyl}piperidin-4-ol
3-({3-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]piperidin-1-yl}methyl)phenol
ethyl 2-(4-{[(1-benzylpyrrolidin-3-yl)carbamoyl]amino}phenyl)acetate