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4-fluoro-N-(2-{[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethyl)benzamide
1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}-1,4-diazepan-5-one
1-(3-methylbutanoyl)-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)piperidine-4-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(3-methoxyphenyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-1-carboxamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-(pyridin-3-yl)acetamide
2-(4-methoxyphenyl)-N-[4-(4-{[2,2,2-trifluoro-1-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
8-[2-(dimethylamino)-2-(3-fluorophenyl)acetyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
methyl 2-[({2-[(2-chloroprop-2-en-1-yl)oxy]-7-fluoroquinolin-3-yl}methyl)amino]-4-(methylsulfanyl)butanoate
[(1-cyclohexylpiperidin-3-yl)methyl]({[5-(methoxymethyl)furan-2-yl]methyl})(pyridin-3-ylmethyl)amine
(3R,4R)-1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
3-(4-hydroxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-pyrazole-5-carboxamide
3-(2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
3-phenyl-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
2-[2-(4-fluorophenyl)azetidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
8-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{[2-chloro-3-(2,3-dihydro-1,4-benzodioxin-6-yloxy)phenyl]methyl}pyrrolidine
7-(cyclohexylmethyl)-2-(6-methylpyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3aR,6aS)-2-ethyl-5-{[(2-fluorophenyl)methyl]carbamoyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(carbamoylmethyl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-4-methylpyrimidine-5-carboxamide
N-[(1R)-1-phenylethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-(dimethylamino)-2-(4-methylphenyl)-N-[2-(pyridin-3-yl)ethyl]acetamide
N-benzyl-N-methyl-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propanamide
8-[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]quinoline
3-(1H-1,3-benzodiazol-2-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
(3aR,5R,6S,7aS)-2-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-octahydro-1H-isoindole-5,6-diol
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-1-methyl-5-phenyl-1H-pyrrole-2-carboxamide
2-(4-hydroxyphenyl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N,N-dimethylpyrazin-2-amine
N-(1-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
7-(3-hydroxy-4-methylbenzoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[2-(4-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1H-1,2,3-triazol-1-yl)ethyl]piperidine
N-(5-chloro-2-methylphenyl)-N'-[1-(pyridin-2-yl)propan-2-yl]propanediamide
3-(3-chlorophenyl)-5-{imidazo[1,2-a]pyrimidine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-(2-methoxyethyl)-1-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-(thiophen-3-ylmethyl)urea
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
4-(naphthalen-2-yloxy)-1-(piperidin-3-ylmethyl)piperidine-4-carboxylic acid
1-(1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-4-yl)piperidin-3-ol
3-cyclopropyl-5-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridin-4-yl}-1H-1,2,4-triazole
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N-ethyl-N-methylpyrimidin-4-amine
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylbenzenesulfonamide
2-{[5-(furan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-3-methylpyridine
1-(4-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}phenyl)pyrrolidin-2-one
2-amino-3-ethyl-N-[2-(2-fluorophenyl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-benzyl-8-(1H-imidazol-4-ylmethyl)-2,8-diazaspiro[5.5]undecane
1-{5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-[4-(2-aminopyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide