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1-(1-methyl-5-{[methyl(quinoxalin-2-ylmethyl)amino]methyl}-1H-pyrrol-3-yl)ethan-1-one
2-(1H-1,3-benzodiazol-2-yl)-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)acetamide
N-(4-methyl-2-oxo-2H-chromen-7-yl)-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
N-{[6-(3,4-dichlorophenyl)pyridin-3-yl]methyl}acetamide
2-(2-phenyl-1,3-thiazol-4-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
1-(2-methoxyethyl)-6-oxo-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine-3-carboxamide
3-(4-methoxyphenyl)-4-[1-(2-methylpropyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
ethyl 3-[(2,4-difluorophenyl)methyl]-1-{[2-(2-hydroxyethoxy)phenyl]methyl}piperidine-3-carboxylate
N-cyclopropyl-1-methyl-3-propyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(thian-4-yl)-2,7-diazaspiro[4.5]decane
(5-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}furan-2-yl)methanol
N,N-dimethyl-3-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)aniline
(3S,4S)-1-[4-(methylamino)pyrimidin-2-yl]-4-(naphthalen-2-yl)piperidin-3-ol
6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-(dimethyl-1,2-oxazol-4-yl)-4-[2,5-dioxo-4-(pyridin-2-yl)imidazolidin-4-yl]piperidine-1-carboxamide
2-{1-[(3-methoxyphenyl)methyl]-4-(9H-purin-6-yl)piperazin-2-yl}ethan-1-ol
(2R,3R)-3-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-cyclopropyl-1-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-4-phenyl-1H-imidazole
{2-[(4aS,7aR)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}urea
{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
6-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-2-methyl-1,3-benzoxazole
2-[(5,6-dimethylpyrimidin-4-yl)amino]hexanamide
2-(4-fluorophenyl)-N-[1-(methoxymethyl)cyclopentyl]imidazo[1,2-a]pyridine-6-carboxamide
4-phenoxy-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxylic acid
N,N-dimethyl-4-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-4-oxobutanamide
5-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1,2-oxazole-4-carboxamide
N-({7-[(4-acetamidophenyl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
5-ethyl-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
4-(4-chlorophenoxy)-1-[(5-methylthiophen-2-yl)methyl]piperidine-4-carboxylic acid
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-2-ethoxypyridine
N-{[1-(hydroxymethyl)cyclopentyl]methyl}-2-(2H-indazol-2-yl)acetamide
N-cyclopropyl-2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]pyridine-4-carboxamide
1-{5-[1-(2-ethoxyacetyl)pyrrolidin-2-yl]thiophene-2-carbonyl}piperidine-4-carboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-(furan-2-yl)-2-oxoacetamide
3-(2H-1,3-benzodioxol-5-yl)-5-(1,2,3,4-tetrahydronaphthalen-2-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-{3-cyclopropyl-1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}-N,N-dimethylpiperidine-1-carboxamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-fluoro-5-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}benzonitrile
6-cyclopentyl-2-methoxy-3-({[6-methyl-2-(methylamino)pyrimidin-4-yl]amino}methyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-chloro-4-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}pyridine
1-(2-fluoro-6-methoxybenzoyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-(2-methoxyphenyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperazin-2-one
N-{2-[4-(dimethylamino)phenyl]ethyl}-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
3-(1-{1-[(2S)-2-aminopropanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea
N-[2-(1H-imidazol-2-yl)ethyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
1-(3-phenyl-1,2,4-oxadiazol-5-yl)-4-(pyrrolidine-1-carbonyl)piperidine