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3-({[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
3-[(4-ethoxyphenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
1-(3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-oxopropyl)pyrrolidin-2-one
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-2-methyl-1-benzofuran-5-carboxamide
3-(2-methyl-1H-indol-1-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]propanamide
2-methyl-4-{3-[3-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}butan-2-ol
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
5-{3-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-3-oxopropyl}-5-[(4-phenylphenyl)methyl]pyrrolidin-2-one
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(prop-2-en-1-yl)piperidine-3-carboxamide
(3S,4S)-1-(benzenesulfonyl)-4-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)amino)pyrrolidin-3-ol
3-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}-1H-indazole
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
3-(3-methoxyphenyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-pyrazole-4-carboxamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-{[2-(trifluoromethoxy)phenyl]methyl}piperidine-3-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-4-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]-1,3-oxazole
N-[(6-chloropyridin-3-yl)methyl]-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methoxybenzoyl)piperazine
2-{1-[(3-phenyl-1H-pyrazol-5-yl)methyl]pyrrolidin-2-yl}-1,3-thiazole
5-(5-methyl-4-phenylthiophen-3-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-methylbut-2-en-1-one
4-(3-hydroxy-3-methylbutyl)-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)benzamide
(1R,5R)-3-(1H-indole-6-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3-methylphenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-({4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1,3-oxazol-2-yl}methoxy)isoquinoline
(1S,5R)-6-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
7-methanesulfonyl-4-methyl-2-{octahydro-1H-pyrido[1,2-a]piperazin-2-yl}quinazoline
1-(carbamoylmethyl)-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]piperidine-4-carboxamide
2-methyl-6-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-yl)-3,4-dihydropyrimidin-4-one
4-hydroxy-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
8-chloro-3-[2-(3,5-dimethylpiperidin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
1-(carbamoylmethyl)-N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
[(5-ethylpyridin-2-yl)methyl](methyl){[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}amine
2-(4-fluorophenyl)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidine
5-(1-ethyl-1H-imidazol-2-yl)-1-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-4-phenyl-1H-imidazole
2-[(2,3,4-trimethoxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
3-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
1-(carbamoylmethyl)-N-(3-hydroxy-3-phenylpropyl)-N-methylpiperidine-4-carboxamide
methyl 3-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}amino)-4-methylbenzoate
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
3-(4-chlorophenyl)-N-(1-ethyl-1H-1,2,4-triazol-3-yl)pyrrolidine-1-carboxamide
6-[(3-methoxyphenyl)methoxy]-4-(5-methyl-1H-pyrazole-3-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-(1,2-oxazol-3-ylmethyl)-3-(trifluoromethyl)pyridin-2-amine
(3S)-3-benzyl-4-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)piperazin-2-one
(1-benzofuran-2-ylmethyl)[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]methylamine