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N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(4-fluorophenyl)-2-hydroxyacetamide
[(2-methylphenyl)methyl](prop-2-en-1-yl)(pyridin-2-ylmethyl)amine
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyridin-2-ylmethyl)piperazine
ethyl 4-({[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}amino)piperidine-1-carboxylate
N-[(3R,4R)-1-[2-(benzyloxy)acetyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(6-methylpyridin-2-yl)methyl]-1-phenylpiperazin-2-one
1-[benzyl(methyl)amino]-3-(5-{[benzyl(methyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
1-(3,4-dimethylphenyl)-5-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-1H-1,2,4-triazole
5-(3-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-3-oxopropyl)imidazolidine-2,4-dione
(1S,5R)-6-(1-methyl-1H-pyrazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
[(3R,4R)-1-(7-fluoro-2-methylquinoline-4-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-(1-hydroxy-3-methylbutan-2-yl)-2-(4-propanoylphenoxy)acetamide
2-(3-{[4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}phenoxy)acetamide
5-ethyl-4-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-methylpyrimidine
N-(pyridin-2-ylmethyl)-4-(quinolin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-methyl-2-[3-(1-propyl-1H-pyrazol-3-yl)phenyl]pyridine
3-amino-N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-1,2,4-triazole-5-carboxamide
2-amino-8-(3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}phenol
2-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}azetidin-3-yl)pyridine
1-(cyclohexylmethyl)-4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-methyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-2-(pyridin-3-yl)acetamide
3-methyl-8-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
(1R,5R)-N,N-dimethyl-6-(3-phenoxypropanoyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-(2-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)phenol
5-{2-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
N-ethyl-2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
1-[(2,3-difluorophenyl)methyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-4-(piperidin-1-yl)butan-1-one
4-[(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methyl]morpholine
2-cyclobutyl-1-[(3R,4S)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]ethan-1-one
4-methoxy-2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenol
3-hydroxy-3-{[(2-phenylethyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-{2-[5-(3,5-difluoro-4-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
N-[5-(1H-pyrazol-3-yl)pyridin-2-yl]methanesulfonamide
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylfuran-2-carboxamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
7-(4-ethylbenzoyl)-2,7-diazaspiro[4.5]decane
1-[(3R,5S)-5-(pyrrolidine-1-carbonyl)piperidine-3-carbonyl]-4-(1,3-thiazol-2-yl)piperazine
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(4-fluorophenyl)-1-[1-(furan-3-ylmethyl)piperidin-4-yl]ethyl]methylamine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N,N,1-trimethyl-1H-1,3-benzodiazole-5-carboxamide
(3R,4S)-3-[3-(1H-1,3-benzodiazol-2-yl)propanamido]-4-cyclopropyl-N,N-dimethylpyrrolidine-1-carboxamide
1-[4-(4-chlorophenoxy)piperidin-1-yl]-2-methyl-3-(morpholin-4-yl)propan-1-one
methyl 3-benzamido-5-{[(2-methoxyphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-chloro-4-[1-(2-methoxyethyl)pyrrolidine-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-4-fluoro-N-(pyridin-3-ylmethyl)benzamide