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N-[(3-{4-[(methylcarbamoyl)amino]phenyl}phenyl)methyl]propanamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
(2S,4R)-1-[(2,6-difluorophenyl)methyl]-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
3-(propan-2-yl)-6-{spiro[2.3]hexan-1-yl}-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
(3aS,6aS)-2-ethyl-5-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-2-(1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)-1H-1,3-benzodiazole
N-{[4-hydroxy-1-(1H-pyrrole-2-carbonyl)azepan-4-yl]methyl}-2-methoxybenzamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-7-fluoro-2-oxo-N-(propan-2-yl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-(2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}pyrimidin-4-yl)piperidin-4-ol
2-methyl-7-(2-phenylbenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(1S,5R)-3-benzyl-6-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-3,6-diazabicyclo[3.2.2]nonane
5-[(2E)-but-2-en-2-yl]-4-phenyl-1-(prop-2-yn-1-yl)-1H-imidazole
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-(2,2-diphenylethyl)-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
4-(4-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
6-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]pyridine-2-carbonitrile
4-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}-5-ethylfuran-2-carboxamide
(2E)-1-[(4aR,8aS)-6-[2-(4-methoxyphenyl)acetyl]-decahydro-1,6-naphthyridin-1-yl]-3-(thiophen-2-yl)prop-2-en-1-one
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[3-(4-fluorophenyl)pyrrolidin-1-yl]ethan-1-one
N-[3-(1H-indazol-1-yl)propyl]-6-methyl-4-oxo-4H-pyran-2-carboxamide
N-methyl-6-(2-phenylpropyl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
{2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-2-oxoethyl}urea
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}cyclohex-3-ene-1-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-benzofuran-5-carboxamide
1-{4-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}ethan-1-one
7,8-dimethyl-4-(piperidine-1-carbonyl)-2-(pyrimidin-5-yl)quinoline
1-{[1-butyl-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]methyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
(5S,9aS,9bS)-5-(3,4-dimethylphenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(2-{[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]formamido}ethyl)piperidine-3-carboxamide
4-(2-hydroxypyridine-3-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
5-(4-benzylpiperidine-1-carbonyl)-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
N-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
(1S,5R)-6-(cyclobutylmethyl)-3-(2-propoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(5-fluoro-2-methylbenzoyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1,4-diazepane-1-carboxamide
N-ethyl-2-(4-propanoylphenoxy)-N-(pyridin-4-ylmethyl)acetamide
2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
7-methyl-2-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
3-(2-amino-1,3-thiazol-4-yl)-1-[3-methyl-4-(propan-2-yl)piperazin-1-yl]propan-1-one
2-(2-methoxyethyl)-9-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-acetyl-8-(5-cyanopyridin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2R,3R,6R)-5-(3-fluoropropyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3R,4S)-N,N-dimethyl-1-(6-methylpyrimidin-4-yl)-4-propylpyrrolidin-3-amine
N-[2-(2-fluorophenyl)-1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N,2-dimethylfuran-3-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(2-methylpropyl)piperidin-4-amine
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2,2-dimethyloxane-4-carboxamide
4-(4-hydroxy-4-methylazepane-1-carbonyl)-1,2-dihydroquinazolin-2-one
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide