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2-[(3,4-difluorophenyl)methyl]-8-{[(2R)-1-methylpyrrolidin-2-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
2-(dimethyl-1,2-oxazol-4-yl)-1-{4-[5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
(1R,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-(2-aminopropanoyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-N'-(4-methylphenyl)propanediamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-indazol-6-amine
N-{4-[(2-methoxyethyl)carbamoyl]-2-methylphenyl}-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]urea
6-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-(3-ethyl-4-methylpiperazin-1-yl)adamantan-1-ol
2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(1R,7S)-3-(4-fluorophenyl)-6-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-[(2-methyl-1H-indol-3-yl)methyl]-2,8-diazaspiro[4.5]decane
4-[4-(dimethyl-1,2-oxazol-4-yl)phenyl]-1,3-thiazol-2-amine
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
(1S,4S)-2-benzyl-5-(1H-1,2,3-triazole-5-carbonyl)-2,5-diazabicyclo[2.2.1]heptane
6-[({[2-fluoro-5-(trifluoromethyl)phenyl]methyl}amino)methyl]-1,4-oxazepan-6-ol
3-methyl-6-(5-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)pyridazine
2-({4-methyl-5-[2-(phenylamino)ethyl]-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-({7-[3-(1,3-benzothiazol-2-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1H-1,3-benzodiazole-2-carboxamide
2-[2-fluoro-6-(propan-2-yloxy)phenyl]pyridine-3-carbonitrile
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
1-[4-(morpholine-4-carbonyl)phenyl]-N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]piperidin-4-amine
3-(3-acetamidophenyl)-4-methylbenzoic acid
(1R,5S,6R)-3-[(1-propyl-1H-imidazol-2-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
2-methyl-6-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]heptan-2-ol
N-(2-{[5-(3-methoxyphenyl)-1,2,4-triazin-3-yl]amino}ethyl)acetamide
(1S,5R)-6-(2-methoxyethyl)-3-[(4-phenylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-(1H-indole-2-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 1-[(3S,5S)-1-(2,2-dimethylpropyl)-5-{[(4-methoxyphenyl)methyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
[(1R,3S,3aS,6aR)-1-(1H-indol-3-ylmethyl)-5-methyl-3-(pyridin-3-yl)-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
8-(4-butylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-fluorophenyl)ethyl]acetamide
N-cyclopentyl-4-(1,4-diazepane-1-sulfonyl)benzamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-methyl-N-[1-(thiophen-2-yl)butyl]-1H-1,2,3-benzotriazole-5-carboxamide
methyl (2S)-1-[5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carbonyl]pyrrolidine-2-carboxylate
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(propan-2-yloxy)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aR)-5-(adamantan-1-yl)-3-[2-(piperidin-1-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-methyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-(2,6-dimethoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[7-(3-fluoro-4-methoxybenzoyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
N-[2-(dimethylamino)ethyl]-8-oxo-7-(prop-2-en-1-yl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
[(3R,4R)-1-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
7-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-2,7-diazaspiro[4.5]decane
1-(2-amino-6-methylpyrimidin-4-yl)-4-(2-hydroxyacetyl)-1,4-diazepane-6-carboxylic acid