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2-methyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
(4aS,8aS)-4a-hydroxy-7-(6-methylpyridazin-3-yl)-N-(propan-2-yl)-decahydro-2,7-naphthyridine-2-carboxamide
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-2-(2-methoxyphenoxy)acetamide
2-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-5-fluoro-N,N-dimethylpyrimidin-4-amine
4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
4-chloro-1-methyl-3-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}-1H-indazole
2-{4-[5,7-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
5-({3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
4-(1H-imidazol-2-yl)-1-(1-methylpiperidine-2-carbonyl)piperidine
2,6,8-trimethyl-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]quinoline-4-carboxamide
2-cyclopentyl-5-[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(6-methylpyridine-2-carbonyl)piperidine-2-carboxamide
3-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyridin-2-one
2-({[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amino}methyl)benzoic acid
2-[1-(2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazol-4-yl)-N-methylformamido]-N-methylpropanamide
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl][(4-fluorophenyl)methyl]methylamine
1-(1-methanesulfonylpiperidin-3-yl)-4-(2-methoxyphenyl)piperazine
{3-[(3-chlorophenyl)methyl]-1-cyclohexylpiperidin-3-yl}methanol
4-chloro-N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}-3-methylbenzamide
2-[4-(azepan-1-ylmethyl)phenyl]-6-(pyridin-2-yl)-3,4-dihydropyrimidin-4-one
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-7-methoxy-1,2,3,4-tetrahydronaphthalen-2-amine
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
4-ethyl-3-[(1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-4-{2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzene-1-sulfonamide
2-({2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzonitrile
N-{[4-(dimethylamino)oxan-4-yl]methyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
4-chloro-5-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-methyl-1H-pyrazole
1-ethyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}ethan-1-one
6-(2-chlorophenyl)-N-(2-hydroxyethyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(3,4-dimethyl-1H-pyrazol-5-yl)-1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propan-1-one
N-[(3S)-1-[7-acetyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidin-3-yl]acetamide
1-cyclohexanecarbonyl-N-[(4-hydroxy-3-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
N-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
N-(1-benzylpyrrolidin-3-yl)-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}propan-1-one
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N,N-dimethylbenzamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-[(5-methylthiophen-2-yl)sulfonyl]-2,8-diazaspiro[4.5]decane
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-[(cyclohexylmethyl)amino]pyrrolidine-2-carboxamide
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-N-(4-sulfamoylphenyl)piperidine-1-carboxamide
N-cyclopropyl-3-{1-[2-(pyridin-2-yl)acetyl]piperidin-3-yl}propanamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-[(3S,4R)-1-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-4-propylpyrrolidin-3-yl]methanesulfonamide
6-methoxy-N,3-dimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1-benzofuran-2-carboxamide
1-(5-ethyl-1,2-oxazole-3-carbonyl)-4-[3-(trifluoromethyl)phenoxy]piperidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}propanamide