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(1S,5R)-6-(cyclopropylmethyl)-3-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(5-methyl-1,3,4-thiadiazol-2-yl)-1-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]urea
5-methanesulfonamido-1-(2-phenylethyl)-N-[1-(pyridin-2-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
4-[(3,4-difluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
7,7-dimethyl-2-(3-phenyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methylpyridin-2-amine
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
1-[(4-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}phenyl)methyl]-1H-1,2,3,4-tetrazole
14-(8-methoxyquinolin-2-yl)-4-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
5-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-N-phenylpyrimidin-2-amine
8-fluoro-6-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
5-[2-(ethylamino)ethyl]-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-one
N-cyclopropyl-3-{[(2-propyl-1,3-thiazol-4-yl)methyl]sulfamoyl}benzamide
2-{3-[(4,4-difluoropiperidin-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}azepan-4-ol
2-cyclopropyl-9-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-amino-N-[(3,4-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-6-methylpyrimidine-4-carboxamide
2-methoxy-5-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}benzoic acid
1-[(4-methoxyphenyl)methyl]-4-(3-phenoxypropanoyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-(1-methylpyrrolidin-2-yl)thiophene-2-carboxamide
6-{4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}pyrazine-2-carboxylic acid
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(dimethylamino)azepan-1-yl]propan-1-one
1-(cyclohexylmethyl)-4-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-1,2,3-triazole
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(5-methylpyridin-3-yl)acetamide
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(propan-2-yloxy)propan-1-one
(1R,5R)-6-benzyl-N-(4-ethylphenyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(3-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propyl)-1H-pyrazole
(1S,4S)-5-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
7-(2-oxoimidazolidin-1-yl)-4-(3-phenyl-1H-pyrazol-4-yl)-1,2,3,4-tetrahydroquinolin-2-one
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(3,4,5-trifluorophenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2-fluorophenyl)methyl]-3-{1-[2-(2-methoxyphenyl)acetyl]piperidin-3-yl}propanamide
(1R,5R)-6-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-methoxy-1-{1'-[2-(morpholin-3-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
(3S,4R)-1-(4-tert-butylbenzoyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
1-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazole
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidine
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
N-[2-(3-methylthiophen-2-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-{[2-chloro-5-methoxy-4-(propan-2-yloxy)phenyl]methyl}-N,N-dimethylpyrrolidin-3-amine
5-ethyl-1'-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aR,7aS)-1-cyclobutanecarbonyl-4-(1,2,4-oxadiazol-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(2,4-difluorophenoxy)ethan-1-one
(5-{1-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol
methyl({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)(pyrimidin-4-ylmethyl)amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
(3S,4R)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(5S)-5-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrrolidin-2-one
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-(methylsulfanyl)acetamide