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4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butanamide
1-{4-[(2-ethylbutyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-methyl-2-(N-methyl-1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
9-(1-ethyl-1H-pyrazole-5-carbonyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopentyl-6-(2-methoxypyridin-3-yl)pyridazin-3-amine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-(1,3-thiazol-4-ylmethyl)pyrrolidine-2-carboxamide
4-[4-(3-chlorophenyl)-1H-1,2,3-triazol-1-yl]-1-(thian-4-yl)piperidine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-{2-[(3-methoxyphenyl)carbamoyl]ethyl}piperidine-1-carboxamide
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(thiophene-2-carbonyl)piperazine
2-[methyl(3-phenylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(2-phenoxypyridin-3-yl)methyl]pyridine-2-carboxamide
2-[3-(5-methylfuran-2-yl)-5-{2-oxo-1-oxaspiro[4.4]nonan-4-yl}-1H-1,2,4-triazol-1-yl]acetic acid
2-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)pyridine-3-carboxylic acid
4-{3-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]phenoxy}-N,N-dimethylpiperidine-1-sulfonamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(1-hydroxybutan-2-yl)-N-[(5-methylthiophen-2-yl)methyl]furan-2-carboxamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-{4-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}acetamide
1-(3-fluorophenyl)-3-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-[1-(4-methyl-2-phenylpyrimidine-5-carbonyl)piperidin-4-yl]piperidin-4-ol
4-[(1-benzothiophen-2-ylmethyl)amino]-N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-[(5-chloro-1H-indol-2-yl)methyl]-2-(methylsulfanyl)acetamide
2-(3-methoxypropyl)-9-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(azepan-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[1-(hydroxymethyl)-9-[(6-methylpyridin-2-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-methoxyethan-1-one
N-[(2-chlorophenyl)methyl]-2-methyl-N-(2-methylpropyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
N-(3-fluorophenyl)-2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]acetamide
(2S)-N-benzyl-1-(piperidin-4-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-2-carboxamide
1-(2-methyl-4-phenylpyrimidine-5-carbonyl)-4-phenylpiperidin-4-ol
3-methyl-7-(5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
[(2S,6S)-4-[(dimethyl-1,2-oxazol-4-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
1-[2-(diethylamino)-2-(furan-2-yl)ethyl]-3-(5-methyl-4H-1,2,4-triazol-3-yl)urea
1-[(5-methylfuran-2-yl)methyl]-4-phenoxypiperidine-4-carboxylic acid
4-({2-[1-(2-methoxy-6-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
(1S,5R)-3-benzyl-6-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonane
2,4-dimethoxy-6-[3-(1H-pyrazol-1-yl)phenyl]-1,3,5-triazine
2-butyl-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-butyl-1-methyl-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperazin-2-one
4-{[5-(2-chlorophenyl)furan-2-yl]methyl}-6-[(5-methyl-1,2,4-oxadiazol-3-yl)methoxy]-1-(propan-2-yl)-1,4-diazepan-2-one
N-(3,4-dimethoxyphenyl)-5-[4-hydroxy-1-(thiolan-3-yl)piperidin-4-yl]-1-benzofuran-2-carboxamide
(3aR,5R,6S,7aS)-2-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-octahydro-1H-isoindole-5,6-diol
9-(2,5-dimethylfuran-3-carbonyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-cyclohexyl-N3-(1-methoxypropan-2-yl)-N5-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
{4-[(4-methoxyphenyl)methyl]-1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}methanol
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-hydroxy-2-methylpropan-2-yl)acetamide
N-cycloheptyl-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
ethyl 3-{[5-(2,5-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}hexanoate
1-(2,3-dihydro-1H-inden-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one