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7-[(3,4-difluorophenyl)methyl]-2-(quinoline-3-carbonyl)-2,7-diazaspiro[4.5]decane
2-amino-1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-2-methylpropan-1-one
1-(2-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
4-[2-(benzyloxy)ethyl]benzamide
5-[4-(2-ethylphenyl)piperazine-1-carbonyl]-4,6-dimethyl-1,2,3,4-tetrahydropyrimidin-2-one
2-hydroxy-1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(4-methoxyphenyl)ethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,1,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-4-yl)quinoline
4-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)-2,1,3-benzoxadiazole
2-{4-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-(morpholin-4-yl)cyclohexane-1-carboxamide
1-{[4-(5-methylfuran-2-yl)phenyl]methyl}-4-(4H-1,2,4-triazol-3-yl)piperidine
2-(3-fluorophenyl)-N-methyl-N-[2-(piperidin-1-yl)ethyl]-1,3-benzoxazole-5-carboxamide
(1R,5R)-3-benzoyl-6-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
ethyl 4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-amido]piperidine-1-carboxylate
N-methyl-N-{[1-(2-methylphenyl)-1H-1,2,3,4-tetrazol-5-yl](phenyl)methyl}pyrazine-2-carboxamide
3-({[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-hydroxyethyl)amino)-1λ6-thiolane-1,1-dione
N-[7-oxo-5-(3-phenylpiperidine-1-carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]thiophene-3-carboxamide
4-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1-(2-methoxyethyl)pyrrolidin-2-one
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1,3-thiazole-4-carboxamide
N-(2-methoxyethyl)-2-[methyl(pyridin-4-ylmethyl)amino]-N-(thiophen-2-ylmethyl)acetamide
N-{1-[(2-chlorophenyl)methyl]-1H-pyrazol-5-yl}-3-propoxypiperidine-1-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}propan-1-one
2,6-dimethoxy-4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenol
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-methyl-4-[1-(5-phenoxyfuran-2-carbonyl)piperidin-4-yl]pyrimidine
9-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecane
N'-{2-[(3-methylpyridin-2-yl)amino]ethyl}-N-(2,4,6-trimethylphenyl)butanediamide
9-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
N-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(4-phenoxyphenyl)methyl]propanamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2,3-dihydro-1-benzofuran-7-carboxamide
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
2-hydroxy-2-(4-methoxyphenyl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]ethan-1-one
2-({4-[4-(3-cyclohexylpyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
4-(5-oxopyrrolidine-3-carbonyl)-1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-1-methyl-1H-pyrazole-4-carboxamide
N-benzyl-N-(3-hydroxy-2-methylpropyl)-3-methylfuran-2-carboxamide
2-(3-fluorophenyl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]azepane
1-(6-cyanopyridin-2-yl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
(3R,4R)-4-cyclopropyl-1-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-3-methylpiperidin-4-ol
N,1,3-trimethyl-2,6-dioxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-benzyl-8-(5-methyl-1,3,4-oxadiazol-2-yl)-2,8-diazaspiro[4.5]decan-1-one
1-cycloheptyl-6-oxo-N-{[2-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-{1-[(3-chloropyridin-4-yl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-{6-oxa-9-azaspiro[4.5]decan-9-yl}butan-1-one
N-{3-[4-({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}(methyl)amino)piperidin-1-yl]phenyl}-4-phenylbutanamide
N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-6-carboxamide
2-({1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(2-methylphenyl)-3-{1-[1-(3-phenylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea