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(3S,4S)-1-(5-chlorofuran-2-carbonyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
1-(3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3aR,7aS)-2-(1-benzyl-1H-pyrazole-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}azetidin-3-ol
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-[(2-methylphenyl)sulfanyl]piperidine
3-(2-methoxyethyl)-1,8-bis(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[(1-cyclohexyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]sulfanyl}pyrimidine
1-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-[1-(2-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]azetidin-3-ol
ethyl 4-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine-1-carboxylate
5-(2H-1,3-benzodioxole-5-carbonyl)-1-ethyl-N-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(3-{[(2-methoxyethyl)amino]methyl}-1H-indol-1-yl)propanamide
4-(5-methylpyridin-2-yl)-1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-4-ol
1-(2-ethoxyethyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
3-cyclohexyl-N-[(1r,4r)-4-hydroxycyclohexyl]-1H-pyrazole-4-carboxamide
2-(1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-4-phenyl-1H-imidazol-5-yl)benzoic acid
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
9-(2-aminopyrimidin-4-yl)-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2,3-dihydro-1-benzofuran-2-carboxamide
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
2-[4-(2-aminopyrimidin-4-yl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(1-benzyl-5-oxopyrrolidin-3-yl)-5-(morpholin-4-ylmethyl)furan-3-carboxamide
5-[(2-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
1-[2-(3-chlorophenyl)ethyl]-4-[(1-methylpiperidin-4-yl)amino]pyrrolidin-2-one
1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-4-(2-propoxyethyl)piperazine
methyl 2-(2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-methylacetamido)acetate
4-[6-(2-methyl-1H-imidazol-1-yl)pyridazin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-({3-methyl-7-[4-(thiophen-2-yl)butanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1H-indole-2-carboxamide
1-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)phenyl]ethan-1-one
N-[(3-chloro-4-fluorophenyl)methyl]-2-methyl-3-[(pyridin-2-ylmethyl)amino]benzamide
7-(2-methoxyethyl)-2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane
2-(4-{[3-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
2-(2-methoxyethyl)-9-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
benzyl 4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,4-diazepane-1-carboxylate
1-(4-phenylpiperazin-1-yl)-3-[1-(quinolin-5-ylmethyl)piperidin-4-yl]propan-1-one
1-[4-(1-cyclopropanecarbonylpiperidin-4-yl)piperazin-1-yl]isoquinoline
1-(3-phenyl-1,2-oxazole-5-carbonyl)-2-(2-phenylethyl)piperidine
N-cyclopropyl-1-[1-(4-methylpentanoyl)piperidin-4-yl]piperidine-3-carboxamide
[(5-ethylfuran-2-yl)methyl]({[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl})amine
2-{4-[1-(isoquinolin-1-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}-N,N-dimethylacetamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-2-hydroxy-4-methylbenzamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-imidazole
(2S)-2-acetamido-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}propanamide
1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]-N-{[4-(morpholin-4-yl)phenyl]methyl}piperidine-4-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
1-cyclopentanecarbonyl-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(3-fluoro-4-methoxybenzoyl)piperidine
[(5-fluoro-1H-indol-2-yl)methyl](methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-(pyrimidin-2-yl)-1,4-diazepane