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(4aS,7aR)-1-butyl-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2,2-diphenylacetamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2,3-dimethyl-1H-indole-7-carboxamide
N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-[1-(dimethylamino)-2-methylpropan-2-yl]-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(3S,4R)-1-[(2-cyanophenyl)methyl]-4-propylpyrrolidin-3-yl]acetamide
5-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-N-propylpyrimidin-2-amine
4-[3-(pyrrolidine-1-carbonyl)phenoxy]-1-(thiolan-3-yl)piperidine
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-5-oxopyrrolidine-3-carboxamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
2-[(4-cyclopentylpyrimidin-2-yl)(methyl)amino]-N-methylacetamide
(3aS,6aS)-2-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2,7-dimethyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-5-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3,5-dimethyl-1-phenyl-1H-pyrazole
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
1-(5-aminopentanoyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
3-(4-hydroxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
7-fluoro-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}quinazolin-4-amine
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzothiazole
2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-3-(thiomorpholine-4-carbonyl)-1,4-dihydropyridin-4-one
1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
(2R,6R)-4-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(phenylsulfanyl)ethan-1-one
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
3-{2-[1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]ethyl}phenol
(2R,4R)-N-[3-(furan-2-amido)-4-methoxyphenyl]-4-hydroxypyrrolidine-2-carboxamide
4-amino-2-{3-[1-(dimethylamino)ethyl]phenyl}pyrimidine-5-carbonitrile
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
4-(1H-pyrazol-3-yl)-1-{[4-(trifluoromethoxy)phenyl]methyl}piperidine
1-(4,6-dimethylpyrimidin-2-yl)-N-[2-(pyridin-2-yl)ethyl]piperidin-4-amine
5-fluoro-2-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]pyridine
(3S,4S)-1-(benzenesulfonyl)-4-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]pyrrolidin-3-ol
methyl (2S,4S)-1-[(4-hydroxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
7-(2-methylphenyl)-4-[2-(pyrrolidin-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(cyclohexylsulfanyl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
methyl 4-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)-1H-pyrazole-3-carboxylate
1-(5-{3-[(3,4-difluorophenyl)amino]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
2-[(1S,5R)-3-[3-(4-fluorophenoxy)propyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-(2-oxopyrrolidin-3-yl)-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
1-cycloheptyl-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-6-oxopiperidine-3-carboxamide
(3R,4R)-3-cyclobutyl-4-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}pyrrolidin-3-ol
methyl 4-{5-[(3-acetamidopyrrolidin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoate
(1R,6S)-N-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
N-{1-[4-(dimethylamino)phenyl]propan-2-yl}-1-(propan-2-yl)piperidine-4-carboxamide
(3R,4S)-1-(2-methoxy-4-methylbenzenesulfonyl)-3,4-dimethylpiperidin-4-ol