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N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-(2-methyl-1H-indol-1-yl)propanamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}piperidin-2-one
2-(cyclopropylmethyl)-N-[(dimethyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-2-ylmethyl)piperidine
4-(6-methoxypyridin-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[2-(1H-imidazol-2-yl)benzoyl]-4-(pyridin-4-yl)piperazine
N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
2-hydroxy-5-{[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]methyl}benzoic acid
(1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(pyridin-3-yl)methanol
1-(4-methylphenyl)-4-(1-phenyl-1H-pyrazole-4-carbonyl)piperazin-2-one
5-({[(4,6-dimethylpyridin-2-yl)methyl](methyl)amino}methyl)-N,N-dimethylpyridin-2-amine
3-(naphthalen-1-ylmethyl)-N-(prop-2-en-1-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)-1H-1,3-benzodiazole
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N,N-diethyl-4-[(1-methylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
2-amino-N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[6-(dimethylcarbamoyl)pyrazin-2-yl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(3S,4R)-4-(4-fluorophenyl)-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]pyrrolidine-3-carboxylic acid
3-(4-methyl-1H-pyrazol-5-yl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
1-(adamantan-1-yl)-4-(1H-pyrrole-2-carbonyl)piperazine
6,7-dimethoxy-3-[1-(pyridin-4-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
1-(2-{methyl[2-(1H-pyrazol-1-yl)ethyl]amino}pyrimidin-4-yl)piperidin-4-ol
5-cyclopropanecarbonyl-1'-[(3-fluoro-2-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(3,4-dimethoxyphenyl)methyl]-2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]acetamide
({4-cyclopropyl-5-[1-(thiophene-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]cyclohexan-1-ol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
(1S,5R)-6-[(2-ethoxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(1R,5R)-6-methyl-N-(4-methylphenyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(methoxymethyl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}cyclobutane-1-carboxamide
4-{4-[(3-chlorophenyl)methyl]piperazine-1-carbonyl}-6-ethyl-1,2-dihydropyridin-2-one
8-(furan-3-ylmethyl)-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(2,3-dihydro-1H-inden-2-yl)-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-cyclopentyl-1H-1,2,4-triazol-5-yl)-2-ethoxypyridine
2-[(4-chlorophenyl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-benzoxazole-5-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-{2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-4-carboxamide
3-chloro-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-(trifluoromethyl)pyridin-2-amine
(cyclopropylmethyl)({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
diethyl({5-methyl-4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]furan-2-yl}methyl)amine
N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
(1R,5S,6R,7S)-3-(2-aminoethyl)-N-[(2,3-dimethylphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
4-[3-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}phenoxy)propyl]morpholine
2-[(2-amino-6-{methyl[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}pyrimidin-4-yl)amino]ethan-1-ol
N-methyl-2-(methylsulfanyl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]acetamide
5-methyl-1'-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(1R,2S,6R,7S)-4-[3-(1,3-thiazole-2-carbonyl)pyridin-2-yl]-4-azatricyclo[5.2.2.02,6]undecane