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N-{2-methyl-3-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]phenyl}furan-2-carboxamide
7-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-[2-(benzyloxy)phenyl]ethan-1-one
2-cyclopropyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
N-[(3-chloro-2-fluorophenyl)methyl]-N-(3-methoxypropyl)-1-methylpiperidin-4-amine
N,N-bis(2-methylpropyl)-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-2-(3-oxopiperazin-1-yl)acetamide
4-hydroxy-1-(4-methoxy-2,3,6-trimethylbenzenesulfonyl)piperidine-4-carboxylic acid
1-(3-{[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}propyl)piperidin-3-ol
2-methyl-5-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
3-{2-[(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]ethyl}-1,3-oxazinan-2-one
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
2-[4-(methylsulfanyl)phenyl]-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
8-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-indole-2-carboxamide
N3-benzyl-N3,N5-dimethyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-(2,3-difluoro-4-methoxyphenyl)-1-[2-(1H-imidazol-4-yl)ethyl]-4-phenyl-1H-imidazole
3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-methylurea
N-(2-methoxyethyl)-2-(5-methyl-1,2-oxazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
N-cyclopropyl-2-(2-fluoro-5-methoxyphenyl)pyridine-4-carboxamide
1-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
4-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(oxan-4-yl)pyridin-2-amine
1'-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
4-[2-(2-methylpropyl)morpholin-4-yl]-N-(pyridin-2-ylmethyl)pyridine-2-carboxamide
5-hydroxy-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pyridine-2-carboxamide
(3S,4S)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-propylpyrrolidine-3-carboxylic acid
2-[2-fluoro-4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
[(2,2-dimethyloxan-4-yl)methyl](ethyl)[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-(5-{[5-(oxan-2-yl)furan-2-yl]methyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
1-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-methylurea
N-[(1R,2R)-2-(dimethylamino)-2,3-dihydro-1H-inden-1-yl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine
2-(4-methoxyphenyl)-5-methyl-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole
N'-cyclopentyl-N-[2-methoxy-2-(thiophen-2-yl)ethyl]butanediamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-methylacetamide
7-propyl-2-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-cycloheptanecarbonylpiperidine
1-[3-(4-ethyl-2-methyl-3-oxopiperazin-1-yl)-3-oxopropyl]azepan-2-one
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
1-(furan-2-carbonyl)-4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
1-[4-(oxolan-2-ylmethoxy)phenyl]-3-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}urea
1-(5-fluoropyridin-3-yl)-3-[1-(furan-2-carbonyl)piperidin-3-yl]urea
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]ethan-1-one
N-(1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
ethyl[2-(1H-pyrazol-1-yl)ethyl][(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide