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4-(1H-imidazol-1-yl)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidine-4-carboxylic acid
ethyl 3-[(2-fluorophenyl)methyl]-1-(oxane-4-carbonyl)piperidine-3-carboxylate
2-(cyclopropylmethyl)-9-[2-(methylsulfanyl)pyrimidine-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
[3-(2-methoxyethyl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]piperidin-3-yl]methanol
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]thiophen-3-amine
2-methyl-N-{2-[7-(3-phenoxypropanoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
N-cyclohexyl-1-ethyl-N-[2-(ethylsulfanyl)ethyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
5-(oxolan-2-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}thiophene-2-carboxamide
1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-N-phenylpiperidin-3-amine
2-{3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
N-[(1-{[2-(2-phenylethynyl)phenyl]methyl}piperidin-3-yl)methyl]furan-2-carboxamide
1-(4-benzylpiperidin-1-yl)-3-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]propan-1-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-propyl-1H-pyrazole-5-carboxamide
6-{1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-3-yl}pyrimidin-4-ol
(3R,5S)-N-[3-(dimethylamino)propyl]-5-(morpholin-4-ylmethyl)-1-(2-phenylethyl)piperidine-3-carboxamide
3-[(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)carbamoyl]pyridin-1-ium-1-olate
2-amino-4-(3-ethoxy-4-hydroxyphenyl)-6-(propan-2-yl)pyridine-3-carbonitrile
4-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyrimidin-2-amine
1-[2-(dimethylamino)-4-{[(2-ethoxypyridin-3-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-(3-ethylphenyl)-4-oxo-4-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]butanamide
1-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-yl]-2-methyl-2-(1H-pyrrol-1-yl)propan-1-one
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(4-fluorophenyl)methyl]piperidine
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]acetamide
(1S,5R)-6-[5-(methoxymethyl)furan-2-carbonyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4-{[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]methyl}phenoxy)-1-(morpholin-4-yl)ethan-1-one
1-(4-{[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]sulfonyl}phenyl)ethan-1-one
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]urea
2-{3-[2-(4-chlorophenoxy)ethyl]phenyl}-5-methyl-1,3,4-oxadiazole
3-(2-methyl-1H-imidazol-1-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1-benzofuran-2-carboxamide
2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carboxylic acid
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-9H-purin-6-amine
3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
4-phenyl-1-[2-(1H-pyrazol-1-yl)butanoyl]piperidine-4-carbonitrile
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)furan-2-carboxamide
1-(propan-2-yl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-{2-[cyclopentyl(methyl)amino]ethyl}-6-ethyl-N,2-dimethylquinoline-4-carboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
3-[2-(2,4-difluorophenyl)ethyl]-1-(2-ethoxyethyl)piperidine
2-amino-6-methyl-N-(5-methyl-2-pentanamidophenyl)pyrimidine-4-carboxamide
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(2-methoxyethyl)methylamine
2-{2-[1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
2-amino-8-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-({1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)cyclopropanesulfonamide
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
2-[3-(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-1H-pyrazol-3-yl)phenyl]pyrazine
N-(1H-imidazol-2-ylmethyl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide