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1-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-methylpiperazine
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]-1H-1,3-benzodiazole
1-{4-[3-(1-hydroxyethyl)phenyl]phenyl}-3-methylurea
5-(dimethylamino)-2-{2-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
1-[(4-chlorophenyl)methyl]-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
4-(2,4-dioxoimidazolidin-1-yl)-N-(furan-3-ylmethyl)-N-methylbenzamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(1H-pyrazol-1-yl)propanamide
4-{2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]-1-(pyridin-2-yl)ethyl}morpholine
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(thiophene-2-carbonyl)piperidine
N-(2,3-difluorophenyl)-3-{[methyl(oxolan-2-ylmethyl)amino]methyl}benzamide
N-[(3,4-difluorophenyl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-decahydro-1,6-naphthyridin-2-one
2-[4-(hydroxymethyl)phenyl]-2-[methyl(1,3-thiazol-2-ylmethyl)amino]acetic acid
1-[1,3-dioxo-2-(quinolin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
3-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-3-yl]propan-1-ol
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)furan-2-carboxamide
(2S)-2-amino-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
1-(2-oxo-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(2R,3R)-1'-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
3-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole
N-(2-methoxy-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)-3-oxo-2,3-dihydro-1H-indene-1-carboxamide
[(3R,4R)-1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}urea
1-(4-phenylpiperazin-1-yl)-3-[1-(thiolan-3-yl)piperidin-4-yl]propan-1-one
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
2-[methyl(pyridin-3-ylmethyl)amino]-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)ethan-1-one
9-(3-hydroxybenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[(5-chloro-2,3-dimethoxyphenyl)methyl]-2-oxopiperazin-1-yl}benzonitrile
1-[(2-chlorophenyl)methyl]-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)butanamide
(3R,4R)-1-(3-methoxypyrazin-2-yl)-3,4-dimethylpyrrolidin-3-ol
5-methyl-3-[1-(pyridin-3-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
8-[6-(piperidin-1-yl)pyrimidin-4-yl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-propyl-5-({2-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidin-2-amine
[1-methyl-5-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
2-(2,4-dichlorophenoxy)-1-[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methyl-1,3-thiazole-5-carboxamide
1-methyl-3-phenyl-4-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
1-(1H-indazol-6-yl)-5-methyl-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-2-one
5-cyclobutyl-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1,3,4-oxadiazol-2-amine
(4-{[methyl({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl})amino]methyl}oxan-4-yl)methanol
methyl 2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxylate