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2,6-difluoro-N-{[7-(thian-4-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
N-[1-(1H-indol-5-yl)ethyl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-2-oxo-4-(1H-pyrazol-3-ylmethyl)-1,4-diazepan-6-yl}oxy)acetamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-[(cyclohexylmethyl)amino]-N-methylpyrrolidine-2-carboxamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-ethyl-7-(2-methoxybenzamido)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N,2-dimethyl-3-[({2-[3-(propan-2-yloxy)phenyl]ethyl}carbamoyl)amino]benzamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
(3S,9aR)-3-(4-aminobutyl)-8-(2-phenylethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-fluoro-N-(2-{3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}ethyl)benzamide
2-[3-(3-methoxyphenoxy)propyl]pyridine-4-carbonitrile
2-(4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}morpholin-3-yl)acetamide
3-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]pyridin-2-ol
N-methyl-2-(2-oxo-1,2-dihydroquinoxalin-1-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
1-[2-(pyridin-2-yl)ethyl]-5-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)piperidin-2-one
diethyl({3-[3-(methoxymethyl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
5-[3-(4-fluorophenyl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
8-(5-phenyl-1,2,4-oxadiazol-3-yl)-1-oxa-8-azaspiro[4.5]decane
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
N-(3-chloro-2-ethoxyphenyl)-3-(morpholin-4-yl)azetidine-1-carboxamide
1-(4-{2-[2-(2-aminoethyl)morpholin-4-yl]-2-oxoethoxy}phenyl)propan-1-one
4-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazine-1-sulfonamide
N-ethyl-5-{[(1R,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyrimidin-2-amine
2-(morpholin-2-yl)-N-propyl-N-(pyridin-3-ylmethyl)acetamide
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-(quinolin-5-yloxy)piperidine-4-carboxamide
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}propan-1-one
(4S,4aS,8aS)-1-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-4-phenyl-decahydroquinolin-4-ol
(1S,5R)-3-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-[(6-methoxynaphthalen-2-yl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
3-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]-1-(thiolan-3-yl)urea
1-methyl-2-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-{[4-(benzyloxy)phenyl]methyl}-4-(2-methoxyethyl)-1,4-diazepan-5-one
1-(3-chloro-4-methylphenyl)-4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}piperidine
(4aS,8aR)-1-(3-methoxypropyl)-6-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-(4-{[(prop-2-en-1-yl)(propan-2-yl)amino]methyl}thiophen-2-yl)ethan-1-one
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(4-methoxy-3-methylphenyl)methyl]piperidine
4-(6-methoxypyridazin-3-yl)benzamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amine
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(1R,2R,6S,7S)-4-(6-methylpyridine-2-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
3-[(3,4-difluorophenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(1-methylpiperidin-2-yl)-1-[4-(pyridin-4-yl)piperazin-1-yl]propan-1-one
3-[2-(pyridin-2-yl)piperidin-1-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}azetidin-3-ol
(1-methoxypropan-2-yl)[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]amine
N-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]acetamide
4-[3-(2-chlorophenyl)pyrrolidin-1-yl]-N-cyclopentyl-4-oxobutanamide
1-cyclobutanecarbonyl-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-methyl-4-[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]-1,4-diazepane
1-acetyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide