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1-methyl-4-[2-(phenylsulfanyl)ethyl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]furan-3-carboxamide
5-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N,5,6-trimethyl-N-(pyridin-3-ylmethyl)-2-(pyrrolidin-1-yl)pyrimidin-4-amine
4-(3-phenyl-1,2,4-oxadiazol-5-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-methyl-4-{2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-oxoethyl}-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
N-[2-(4-ethylphenyl)ethyl]-2-(morpholin-2-yl)acetamide
5-(5-chloro-2-methoxypyridin-4-yl)-2,4-dimethoxypyrimidine
4-methyl-13-(3,3,3-trifluoropropyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
[(3R,4S)-1-[(4-fluoro-3-methoxyphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-amino-5-methyl-4-[5-(1H-pyrazol-3-yl)furan-2-yl]-6-(pyridin-2-yl)pyridine-3-carbonitrile
(3S,4S)-1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
4-phenyl-1-[6-(thiomorpholin-4-yl)pyridine-3-carbonyl]azepane
2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]acetamide
(3S,4S)-1-(morpholine-4-sulfonyl)-4-propylpyrrolidine-3-carboxylic acid
ethyl 4-(2-phenylethyl)-1-(pyridin-2-ylmethyl)piperidine-4-carboxylate
2-(ethoxymethyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-methoxy-N-{1-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
4-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-N-(1,2,3-thiadiazol-5-yl)benzamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-(propan-2-yl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
3-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
ethyl 2-(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
N-butyl-2-cyclobutaneamido-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
2-(3-{1-[4-(2-hydroxyethyl)phenyl]-1H-imidazol-2-yl}phenoxy)ethan-1-ol
2-(azocan-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
2-methanesulfonyl-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
8-(1,3-benzoxazol-2-yl)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,8-diazaspiro[4.5]decane
N-methyl-3-(piperidin-3-yl)-N-[2-(pyridin-2-yl)ethyl]benzamide
1-[2-({[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-methyl-N-[2-(pyridin-2-yl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(3aR,6aR)-2-methanesulfonyl-N-[2-(2-oxopyrrolidin-1-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
5-acetyl-N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N,2,4-trimethyl-1H-pyrrole-3-carboxamide
N,N-dimethyl-3-[2-({methyl[1-(1,3-thiazol-2-yl)ethyl]carbamoyl}amino)phenyl]propanamide
1-[5-(4-methoxyphenyl)furan-2-carbonyl]-4-(2-methylpropyl)-1,4-diazepan-5-one
9-(1,2,4-oxadiazol-3-ylmethyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-phenyl-1,2-oxazole-3-carboxamide
2-(2-chlorophenyl)-3-methyl-N-[2-(propan-2-yloxy)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-{4-[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]piperidin-1-yl}ethan-1-one
N-cyclopentyl-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)acetamide
2-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
4-[(dimethylamino)methyl]-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]azepan-4-ol
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
(1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidin-4-yl)(thiophen-2-yl)methanol
N-ethyl-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)-N-propylbenzamide
3-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
3-[4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]propan-1-ol
(4aS,8aR)-6-(4-methylpiperazine-1-carbonyl)-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one