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(2-{2-[1-(3-fluoro-4-methoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2-(1H-pyrazol-1-yl)-N-[2-(pyrrolidin-1-yl)ethyl]butanamide
1-(azocan-1-yl)-3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}propan-1-one
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)piperidine-3-carboxamide
6-methyl-5-{5-[3-(thiophen-2-yl)propyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
2-(2,3-dihydro-1H-inden-2-yl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-methyl-N-{1-[1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-4-yl]-2-phenylethyl}pyridine-2-carboxamide
1-(oxan-4-yl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
5-[1-(4-methoxyphenyl)-1H-pyrazol-3-yl]-4-methyl-N-(thiophen-2-ylmethyl)-1,3-thiazol-2-amine
3-(methoxymethyl)-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
5-ethyl-3-({2-[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)cyclopentanecarboxamide
5-ethyl-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,2-oxazole-3-carboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
4-({9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}methyl)benzonitrile
1-[(4-fluorophenyl)methyl]-4-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4-diazepane
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
7-amino-N-[(1R,3R)-3-aminocyclopentyl]-2-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
4-(1H-indazol-6-yl)-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
2-methyl-4-{3-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]phenyl}but-3-yn-2-ol
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(1H-pyrazol-1-yl)butanamide
1-[3-(methylsulfanyl)propyl]-4-phenyl-1,4-diazepane
2-[4-(3-fluorophenyl)-1H-pyrazol-1-yl]-N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
3-(5-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-[(4-methylpiperazin-1-yl)methyl]piperidin-2-one
N-ethyl-2-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}pyrimidin-4-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(morpholin-3-yl)acetamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(5-methylpyrazine-2-carbonyl)piperidine-4-carboxylic acid
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2,6-dimethoxypyridine-3-carboxamide
1-{1-[3-(2-methyl-1,3-thiazol-4-yl)-1-phenyl-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
N,3,5-trimethyl-N-[1-(pyridin-3-yl)pentyl]-1H-indole-2-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-methyl-1,3-thiazole
1-phenyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-1,2,3-triazole-5-carboxamide
2-(3,4-difluorophenyl)-5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl][1-(1H-pyrazol-1-yl)propan-2-yl]amine
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(3-chloro-1,2-oxazol-5-yl)propan-1-one
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-3-(1H-pyrazol-1-yl)propanamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(thian-4-yl)piperidin-4-yl]acetamide
4-({1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}oxy)-3-chloro-N-(2-methoxyethyl)benzamide
4-{[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-2-methoxyphenol
N-[2-(1H-imidazol-4-yl)ethyl]-2-(naphthalen-2-yloxy)propanamide
(1R,2R,4R)-N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperazin-2-one
N-[2-(dimethylamino)ethyl]-3-{1-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-yl}propanamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]propan-1-one
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(3-methylthiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(1-benzylpyrrolidin-3-yl)amino]-N-(2,3-dimethylphenyl)acetamide
1-[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
1,4-dimethyl-9-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecane
5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(thiophen-3-ylmethyl)-1,2,4-oxadiazole