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1-(2-fluorophenyl)-4-[(3-{[1-(pyridine-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-N'-(2-methylphenyl)propanediamide
N-[4-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenyl]acetamide
N-(1,4-dioxan-2-ylmethyl)-6-(2-methoxyphenyl)pyridazin-3-amine
6-(2-methoxyphenyl)-N-(3-methoxypropyl)pyridazin-3-amine
1-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
2-{4-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
3-tert-butyl-1-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
8-[2-hydroxy-5-(1H-pyrrol-1-yl)benzoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-(2-fluorophenyl)-N-(oxolan-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
3-{[(2-methoxyethyl)(propan-2-yl)amino]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
2-[(2-fluorophenyl)methyl]-4-(4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
[4-(1-benzothiophen-7-yl)pyridin-2-yl]methanol
N-tert-butyl-1-cyclohexyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-cyclopentyl-3-{[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]sulfamoyl}benzamide
1-cyclopentanecarbonyl-N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
(4aS,7aR)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{2-[1-(3,4-difluoro-5-hydroxyphenyl)-1H-imidazol-4-yl]ethyl}acetamide
N-butyl-4-{[2-(2-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
6-acetyl-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
methyl 1-ethoxy-8-(1H-indazole-3-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(2-hydroxyethyl)-2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
{3-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-oxopropyl}urea
2-(4-chlorophenyl)-4-[1-(2-methoxyethyl)piperidine-4-carbonyl]morpholine
N-methyl-4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-amine
3-(2-aminoethyl)-4-[4-chloro-3-(trifluoromethyl)phenyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(quinolin-6-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
N-({3-[(dimethylamino)methyl]phenyl}methyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(furan-2-yl)ethane-1,2-dione
(2S,4R)-4-(4-{4-[(4-hydroxypiperidin-1-yl)methyl]phenyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]furan-2-carboxamide
2-(benzyloxy)-1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-[4-(adamantan-2-yl)-1-benzylpiperazin-2-yl]ethan-1-ol
(1-benzofuran-2-ylmethyl)(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-{1-azabicyclo[2.2.2]octan-3-yl}-6-chloro-2-methylquinoline-4-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-{1,9-dioxaspiro[5.5]undecan-4-yl}propanamide
(1R,5R)-6-(cyclobutylmethyl)-3-(3,5-dimethylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
8-chloro-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]quinoline-2-carboxamide
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
2,6-dimethyl-4-({[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]amino}methyl)phenyl acetate
2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carboxamide
3-({2-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2,4-trimethylpyrimidine-5-carboxamide
{2-[(1S,4S)-5-(2-methoxy-5-phenylphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-oxoethyl}urea
2-ethyl-9-(quinoline-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-(propan-2-yl)piperidine-3-carboxamide
[(2S,6S)-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-tert-butyl-6-[(3-hydroxybutyl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-ethyl-5-({3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}methyl)pyrimidine