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3-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-1-[2-(pyridin-3-yl)ethyl]urea
5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-N-(2-phenylethyl)pyrimidin-2-amine
3-{2-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidin-1-yl)-3-phenylpropan-1-one
1-(oxolan-2-ylmethyl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
4-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]thiomorpholine
3-(1-butyl-1H-pyrazol-5-yl)-1-{[4-(piperidine-1-carbonyl)phenyl]methyl}urea
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-2-(trifluoromethyl)benzamide
2-(2-oxo-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-4-phenyl-1,2-dihydrophthalazin-1-one
1-[4-(ethylamino)pyrimidin-2-yl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
(1S,5R)-6-(2,4-dimethylpyrimidine-5-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-({3-[(3-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-3-methoxypyrrolidine
2-methyl-4-phenyl-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]pyrimidine
9-[(1-ethyl-1H-pyrazol-3-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-5-methyl-3,4-dihydroquinazolin-4-one
3-{[1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)(2-methylpropyl)(pyridin-2-ylmethyl)amine
3-[3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3-chloropyridin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(2-methylphenyl)-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
2-(ethoxymethyl)-N-[(1-propyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl(1-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-2-phenylethyl)(pyridin-4-ylmethyl)amine
2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-1-cyclopentanecarbonylpiperidine-4-carboxamide
1-(furan-3-carbonyl)-4-[3-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepane
(3aR,6aR)-2-(2,3-difluorobenzoyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{9-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
1-[(5-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]azepane
(2S,4S)-4-(3-chlorobenzamido)-1-methyl-N-[3-(methylsulfanyl)propyl]pyrrolidine-2-carboxamide
3-(3-methoxyphenyl)-4-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1H-pyrazole
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[6-(piperidin-3-yl)pyrimidin-4-yl]piperazin-2-one
(1S,5R)-3-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyridin-2-amine
1-(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(phenylsulfanyl)ethan-1-one
methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
(2-{2-[1-(5-chlorothiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2-(dimethylamino)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-2-(4-methylphenyl)acetamide
1-(2-aminoethyl)-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]-5-methoxy-1,4-dihydropyridin-4-one
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-(2-phenylethyl)piperidin-4-amine
1-(3,5-difluoropyridine-2-carbonyl)azepan-3-amine
1-[2-({[2-(pyrrolidin-1-yl)ethyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-{1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]piperidin-4-yl}piperidin-3-ol
4-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}thiomorpholine
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
5-{1-[3-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazol-2-yl}thiophene-2-carboxylic acid
2-(cyclopropylmethyl)-8-(2-methyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one