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[(2,6-difluorophenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-(4-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}piperidin-1-yl)butan-1-one
3-{3-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propyl}pyridine
5-methyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
1-[4-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
(2S,4R)-4-{[(2,6-difluorophenyl)methyl]amino}-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
5-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-ethyl-3-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazole
2-{[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]methyl}benzoic acid
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-2,4-dimethylpyrimidine-5-carboxamide
1-(cyclohexylmethyl)-4-{[(3-hydroxy-4-methoxyphenyl)methyl]amino}pyrrolidin-2-one
5-(propan-2-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1,2-oxazole-3-carboxamide
3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
4-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]benzamide
N-[1-(1H-1,2,4-triazol-5-yl)ethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-[3-(4-ethyl-2-methyl-3-oxopiperazine-1-carbonyl)phenyl]cyclopentanecarboxamide
N,N-dimethyl-7-(1-methylpyrrolidine-3-carbonyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{3-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethylpyridine-3-sulfonamide
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
5-chloro-N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
5-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-2-methylpyrimidine
1-(2-{imidazo[1,2-a]pyridin-3-yl}acetyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(azepane-1-carbonyl)-5-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-1-(2-methylpropyl)-1,4-dihydropyridin-4-one
N-[(3S,4R)-1-(2-phenylacetyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-(carbamoylamino)-N-[(3R,4S)-1-(6-cyclopropylpyrimidin-4-yl)-4-propylpyrrolidin-3-yl]acetamide
(4aS,7aR)-1-[2-(3,4-dimethylphenoxy)acetyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4-methylphenyl)methyl]-5-oxo-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrrolidine-3-carboxamide
[(4-{2-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
3-(2-fluorophenyl)-5-[5-(methoxymethyl)thiophene-2-carbonyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2,3-difluoro-6-methoxybenzamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(2,3-difluoro-4-methoxybenzoyl)piperidine
1-[1-(isoquinolin-4-yl)-1H-pyrazol-3-yl]ethan-1-one
(4aS,8aR)-6-[2-(1H-indol-1-yl)acetyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
1-cyclopentyl-4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-2-one
1-(2,3-dihydro-1H-inden-2-yl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(4-acetyl-4-phenylpiperidin-1-yl)-4-(1H-pyrazol-4-yl)butan-1-one
2-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrido[2,3-d]pyrimidin-4-amine
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-[2-(diethylamino)ethyl]-N-ethylpropanamide
9-[2-hydroxy-2-(4-methoxyphenyl)acetyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-fluorophenyl)methyl]-N-(1-phenylethyl)-2-(1H-pyrazol-1-yl)acetamide
1-[(4-methoxypiperidin-1-yl)sulfonyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-1-carboxamide
3-(1H-1,3-benzodiazol-1-yl)-N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]propanamide
3-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-3,9-diazaspiro[5.6]dodecan-10-one