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9-[2-(4-fluoro-3-methylphenyl)acetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-2-one
ethyl 3-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]amino}propanoate
(3S,4S)-4-(pyridin-2-yl)-1-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidine-3-carboxylic acid
4-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
2-[7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-4-carboxamide
(4aS,7aR)-1-[2-(2-fluorophenyl)acetyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,6R)-N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
N-(4-{4-[(1H-indol-2-ylmethyl)amino]piperidin-1-yl}phenyl)benzenesulfonamide
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1-oxo-2-[2-(pyridin-4-yl)ethyl]-2,3-dihydro-1H-isoindole-5-carboxamide
4-({2-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
(3aS,6aS)-2-(1,3-benzothiazol-2-yl)-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[4-({[2-(3-chlorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
3-(cyclopropylmethyl)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxylic acid
1-(2,6-dimethylpyridine-4-carbonyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1-methylcyclopropyl)propan-1-one
5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-phenyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
1-[(1-{6-[3-(hydroxymethyl)pyrrolidin-1-yl]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(1R,5R)-3-(pyridine-3-carbonyl)-6-(1,3-thiazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
9-[(2S)-2-aminohexanoyl]-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-2-carbonitrile
1-(2-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}pyrrolidin-1-yl)propan-1-one
3-ethyl-8-(oxolan-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-benzyl-1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-one
N-methyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1-methylpiperidin-4-yl)acetamide
(3S,4R)-4-(2-methoxyphenyl)-1-(6-methylpyridine-2-carbonyl)pyrrolidine-3-carboxylic acid
3-[5-(4-methylphenyl)furan-2-yl]-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]propanamide
8-(1-hydroxypropan-2-yl)-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(dimethyl-1,3-oxazole-4-carbonyl)-3-(3-methoxyphenoxymethyl)piperidine
ethyl 1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-ethyl-3-(2-methylpropyl)-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
(3S,5R)-N3-[(3,4-dimethoxyphenyl)methyl]-N5-(4-fluorophenyl)-1-(naphthalen-2-ylmethyl)piperidine-3,5-dicarboxamide
(2S,4S)-N,N-diethyl-4-(2-fluorobenzamido)-1-(3-methylbut-2-en-1-yl)pyrrolidine-2-carboxamide
(3R,4R)-3-methyl-1-[2-(methylamino)pyrimidine-5-carbonyl]-4-(oxan-4-yl)piperidin-4-ol
2-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
5-fluoro-2-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]-1H-1,3-benzodiazole
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline-4-carboxylic acid
2-[2-(4-fluorophenyl)piperidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
5-[(1,3-benzothiazol-2-ylmethyl)amino]-1-methyl-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(5-hydroxyadamantan-2-yl)-5-methyl-4-{[(5-methylfuran-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
({4-[1-(2-methoxypyridine-3-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
4-(2-methylphenoxy)-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid
2-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-S-(4-fluoro-3-methylphenyl)-2-oxoethane-1-sulfonamido
(1R,5S)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonane
2-(2-methyl-1,3-thiazol-4-yl)-5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl){8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}amine
N-[2-(2-fluorophenyl)-1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)ethyl]-N-methylthiophene-2-carboxamide