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2-[(4-chlorophenyl)methyl]-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-[(6-methylpyridin-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
[2-(2H-1,3-benzodioxol-5-yl)ethyl](methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
5-({3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-2,1,3-benzothiadiazole
2-amino-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}acetamide
N4-[3-(dimethylcarbamoyl)-2-methylphenyl]-N1,N1-dimethylpiperazine-1,4-dicarboxamide
2-(piperidin-1-ylmethyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)-1,4-oxazepane
2-({2-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
3-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
4-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
[(3R,4R)-1-(3-aminothiophene-2-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-2,7,8-trimethylquinoline-4-carboxamide
ethyl 1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine
1-(1-methoxypropan-2-yl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-(2,2-dimethyloxan-4-yl)-1-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[(1-ethyl-1H-imidazol-5-yl)methyl]benzamide
9-(2,3-dihydroxybenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(dimethylamino)-1-phenylpropyl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
4-{2-[3-(2-methylphenyl)piperidin-1-yl]pyridine-4-carbonyl}morpholine
5-(methoxymethyl)-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}thiophene-2-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(1,1-dioxo-1λ6-thian-4-yl)acetamide
(3aS,6aR)-3-cyclopentyl-5-(isoquinolin-1-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(3-fluorophenyl)-6,6-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
6-ethyl-2-methyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]quinoline-4-carboxamide
5-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-oxopentanamide
2-[({[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}amino)methyl]-3,4-dihydroquinazolin-4-one
1-[(1S,5R)-6-(2,8-dimethylquinoline-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
4-(5-chloro-3-phenyl-1H-indole-2-carbonyl)piperazine-2-carboxylic acid
5-methyl-2-[1-(oxolane-3-carbonyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-yl]pyridine
2-(2-fluorophenyl)-N-[2-(thiophene-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]acetamide
1-benzyl-N,N-dimethyl-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{2-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-(4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazin-1-yl)-3-methylpyrazine
4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-6-hydroxy-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
2-methoxy-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
methyl 1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decane-8-carboxylate
2-{1-[(2-fluorophenyl)methyl]-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
N-[2-(2-hydroxyethoxy)ethyl]-3-(4-methylphenyl)-3-phenylpropanamide
(2S,4S,5R)-4-[(carboxymethyl)carbamoyl]-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
1-(2,5-dimethylfuran-3-carbonyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)imidazo[1,2-a]pyrimidine-2-carboxamide