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3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]urea
2-[6-(methoxymethyl)pyrimidin-4-yl]-1-methyl-1H-indole
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-(3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
(1R,3S)-N,N,2,2,3-pentamethyl-3-[3-(pyridin-3-yl)azetidine-1-carbonyl]cyclopentane-1-carboxamide
2-(methylamino)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}pyrimidine-5-carboxamide
(2S,4R)-N-ethyl-1-(furan-3-ylmethyl)-4-[3-(5-methyl-1H-pyrazol-1-yl)propanamido]pyrrolidine-2-carboxamide
N-benzyl-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-[(1R,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-benzylacetamide
N-[1-(4-fluorophenyl)ethyl]-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-(1H-imidazol-1-ylmethyl)-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide
N-[(4-tert-butylphenyl)methyl]-5-ethyl-1,3,4-oxadiazol-2-amine
4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-methyl-5-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}pyrrolidin-2-yl)-1,2-oxazole
N-methyl-N-[(4-phenoxyphenyl)methyl]-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-4-carboxamide
(1S,5R)-3-[2-(2,6-dimethoxyphenoxy)ethyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-2-amine
5-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2-methoxyphenol
(1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)(pyridin-2-yl)methanol
1-{[3-(4-methanesulfonylphenyl)phenyl]methyl}piperazine
N,N-dimethyl-2-[({7H-pyrrolo[2,3-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-methyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)furan-2-carboxamide
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-methoxy-3-{thieno[2,3-d]pyrimidin-4-yl}pyridine
(3S,4R)-1-(6,8-dimethoxy-4-methylquinolin-2-yl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
3-[2-(2,6-difluorophenyl)ethyl]-1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidine
N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)cyclohexanecarboxamide
1-[(2R,3R)-1'-(cyclopropylmethyl)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1,4-diazepan-5-one
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[(2-methoxy-3,5-dimethylphenyl)methyl]pyrrolidin-3-yl]methanol
5-ethyl-5-[1-(3-methylpyridine-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(3-methyl-1,2-oxazol-5-yl)acetamide
8-(3-hydroxybenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-1-(pyrrolidin-1-yl)cyclohexane-1-carboxamide
N-(2-{[(2-fluorophenyl)methyl]sulfanyl}phenyl)-3-methoxypiperidine-1-carboxamide
N-butyl-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
1-(2-methylphenyl)-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,4-diazepane
(3S,4S)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
1-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-2-methyl-1,4-diazepan-5-one
2-(1,2-benzoxazol-3-yl)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
N-[(1-benzylpyrrolidin-3-yl)methyl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-amino-7-[(2S)-2-phenylbutanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
N-{1-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
3-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-(2-methyl-1-benzofuran-5-yl)urea
N2-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-N1-(pyridin-3-yl)ethane-1,2-diamine
N,N-dimethyl-5-{[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]methyl}furan-2-carboxamide
5-cyclopropanecarbonyl-1'-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]