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4-cyclobutyl-N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-6-methylpyrimidin-2-amine
3-[5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
6-(3-oxo-3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}propyl)-2,3,4,5-tetrahydropyridazin-3-one
ethyl 1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-N-[(2-fluorophenyl)methyl]acetamide
2-(2H-1,3-benzodioxol-5-yl)-5-(1H-pyrazol-3-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
(3aR,6aR)-2-(2-aminopyrimidin-4-yl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}-2-methylpyrimidin-4-ol
ethyl 4-{2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
2,5-dimethyl-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[2-(N-methylmethanesulfonamido)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
1-[4-({[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]imidazolidin-2-one
2-cyclopropyl-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-cyclopentyl-2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
5-[({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]-2-methoxyphenol
2-cyclopropyl-5-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-3,4-dihydropyrimidin-4-one
1-(3,4-diethoxybenzoyl)-4-(1H-imidazol-2-yl)piperidine
1-(furan-3-ylmethyl)-4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-methyl-N,3-bis(propan-2-yl)-1H-pyrazole-5-carboxamide
9-(2-cyclopropylpyrimidine-5-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}pyridine
N'-[2-(propan-2-yl)phenyl]-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]butanediamide
4-chloro-1-methyl-3-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-1H-pyrazole
2-(5-fluoro-2-methyl-1H-indol-3-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}acetamide
N-(1,2-oxazol-3-ylmethyl)-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
N-[(1R)-2-hydroxy-1-phenylethyl]-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
7-(5-fluoro-3,8-dimethylquinolin-2-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
[(5-ethylpyridin-2-yl)methyl]({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
2,3,5-trimethyl-N-[2-(1-methyl-1H-pyrrol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-methyl-4-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}piperazine
8-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(4aS,8aR)-6-(2-amino-6-methylpyrimidin-4-yl)-1-[3-(methylsulfanyl)propyl]-decahydro-1,6-naphthyridin-2-one
N4-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N2,N2,N4,5,6-pentamethylpyrimidine-2,4-diamine
2-methoxy-3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
5-{1-[2-(2-methoxyphenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
3-(1H-1,3-benzodiazol-2-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
[(2-ethoxy-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)methyl]dimethylamine
(3S,5R)-1-[(4-hydroxy-3-methylphenyl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
4-{3-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
2-(dimethyl-1,2-oxazol-4-yl)-N-[3-(methylsulfamoyl)phenyl]pyrrolidine-1-carboxamide
5-amino-4-chloro-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
5-({2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}methyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
methyl 6-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}-3-cyclopropaneamidothieno[2,3-b]pyridine-2-carboxylate
5-acetyl-3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
1'-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-(adamantan-2-yl)-6-{[4-(hydroxydiphenylmethyl)piperidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}-N-(pyrazin-2-yl)acetamide
1-{3-[1-(4-chlorophenyl)cyclopentyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-ethoxyethan-1-one