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[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
(1R,5R)-6-[3-(dimethylamino)benzoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
N-[(1S,2R)-2-{[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]amino}cyclobutyl]methanesulfonamide
1-(azepan-1-yl)-4-[3-(2-methoxyphenoxy)azetidin-1-yl]butane-1,4-dione
5-[(3R,5S)-3,5-bis(hydroxymethyl)piperidine-1-carbonyl]-2-fluorophenol
{4-[(2-chlorophenyl)methyl]-1-(quinoxalin-2-yl)piperidin-4-yl}methanol
2-amino-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
6-ethyl-2-methyl-4-(thiomorpholine-4-carbonyl)quinoline
2-(2-methoxypyridin-3-yl)-6-methylpyridine-3-carbonitrile
4-{imidazo[1,2-a]pyridin-2-ylmethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[(4-ethoxypiperidin-1-yl)methyl]-6-fluoroquinolin-4-ol
N-[3-(1H-indazol-1-yl)propyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-N-[(2-fluorophenyl)methyl]acetamide
N-(pyridin-3-ylmethyl)-3-{[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1,9-dioxaspiro[5.5]undecan-4-amine
(1S,5R)-3-(2-amino-6-methylpyrimidin-4-yl)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 4-{5-[(3-benzoylpiperidin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoate
2-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-azaspiro[4.4]nonan-3-one
(1S,5R)-6-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
6-{[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-methyl-2-{[(2-methylpyridin-4-yl)methyl]amino}pyridine-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-[2-(4-sulfamoylphenyl)ethyl]propanamide
2-{2-[1-(2-oxo-2-phenylacetyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
3-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-1-[4-(1H-pyrazol-1-yl)phenyl]urea
7-amino-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[3-(morpholin-4-yl)propyl]amine
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-[2-methyl-2-(morpholin-4-yl)propyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(2,3-dimethoxyphenyl)methyl]-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]piperazin-2-one
N-(4-cyano-2-ethylphenyl)-4-(2,6-dimethylpyridin-4-yl)piperazine-1-carboxamide
3-({[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}amino)-2,2-dimethylpropan-1-ol
1-(carbamoylmethyl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-4-carboxamide
2-[(1S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1H-1,3-benzodiazole-6-carboxylic acid
(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}piperidin-2-yl)methanamine
[1-(5-ethyl-2-methylpyrimidin-4-yl)-3-[(2-fluorophenyl)methyl]piperidin-3-yl]methanol
2-{[(4-fluorophenyl)methyl](methyl)amino}-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
2-methyl-N-(4-{methyl[2-(2-methylpiperidin-1-yl)ethyl]carbamoyl}phenyl)furan-3-carboxamide
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
5-methyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1,3-oxazole-4-carboxamide
2-[5-(4-phenyl-1,4-diazepane-1-carbonyl)-1H-pyrazol-3-yl]phenol
4-(1H-1,3-benzodiazol-1-yl)-1-(2-cyclopropylacetyl)piperidine-4-carboxylic acid
(1R,5R)-6-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(2-{3-methyl-4-[(4-methylpiperazin-1-yl)methyl]-1H-pyrazol-1-yl}ethyl)piperidine-3-carboxamide
N-(2-ethoxyphenyl)-3-{8-methyl-2,8-diazaspiro[4.5]decan-2-yl}-3-oxopropanamide
6-methoxy-1-methyl-2-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1H-indole
2-ethoxy-5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}pyridine
4-[2-(propylsulfanyl)phenyl]-4H-1,2,4-triazole
N-{3-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]-2,5-dimethyl-1H-pyrrol-1-yl}acetamide