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5-butyl-4-(4-methyl-1H-imidazole-2-carbonyl)-1-(3-phenylphenyl)piperazin-2-one
[3-(2-methoxyethyl)-1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-3-yl]methanol
1-methyl-4-{1-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
8-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{furo[3,2-c]pyridin-4-yl}-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
8-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N4-ethyl-N2-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-2,4-diamine
2-{3-[(3,4-dimethylpiperazin-1-yl)methyl]phenyl}-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
7-[(2,3-difluorophenyl)methyl]-2-propyl-2,7-diazaspiro[4.5]decane
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylazepane-2-carboxamide
2-amino-6-(2,5-dimethylfuran-3-yl)-4-[3-(2-hydroxyethoxy)phenyl]pyridine-3-carbonitrile
9-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3,9-diazaspiro[5.6]dodecane
N-(1-benzylpiperidin-3-yl)-2-cyclobutyl-5-(2-methoxyacetamido)-1-methyl-1H-1,3-benzodiazole-7-carboxamide
N-(furan-2-ylmethyl)-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
2-[(2-chlorophenyl)methyl]-4-{4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-{2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}acetamide
4-[4-(1,2-oxazolidine-2-carbonyl)phenoxy]-1-(2-phenylethyl)piperidine
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](ethyl){[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}amine
7,7-dimethyl-2-[2-(1H-pyrazol-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
[1-(quinolin-3-yl)-1H-1,3-benzodiazol-2-yl]methanol
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
(1R,3S)-3-methoxy-7-(4-methoxyquinoline-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
5-fluoro-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidine
(4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-3-(1,2-oxazinan-2-yl)propanamide
N-(propan-2-yl)-2-(4-{3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanoyl}piperazin-1-yl)acetamide
(4aR,7aS)-1-{2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-1-(5-ethylthiophene-2-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
8-(5-chloro-2,3-dihydro-1H-indole-2-carbonyl)-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(adamantan-1-yl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-[(4-phenylphenyl)methyl]acetamide
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]pyrrolidin-3-yl]urea
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
3-hydroxy-1-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
1-({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)piperidine-4-carboxamide
2-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-2-oxo-N-(1,3-thiazol-2-yl)acetamide
(3aR,7aS)-2-[4-(4-methylphenoxy)piperidine-4-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-methoxy-2-{[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3,5-dimethylpyridine
3-(4-chlorophenyl)-5-(propan-2-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(3R,9aR)-8-(4-ethylbenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
2-(pyridin-4-yl)-7-(4,4,4-trifluorobutanoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)cyclopentanecarboxamide
N-methyl-N-(1-methylpiperidin-4-yl)-3-{1-[(4-phenylphenyl)methyl]piperidin-3-yl}propanamide
dimethyl({[4-methyl-5-(1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
3-[5-(diethylamino)pentan-2-yl]-1-(6-methylpyridin-3-yl)urea
4-(3-hydroxynaphthalene-2-carbonyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
N,N-dimethyl-5-(1-{[(1-methyl-1H-indazol-3-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)thiophene-2-carboxamide
5-methyl-1-({4-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenyl}methyl)-1H-1,2,3,4-tetrazole
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-acetamidobenzamide